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1-ethyl-N-[3-(pyridin-4-yl)propyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
{[5-(2-benzylmorpholine-4-carbonyl)furan-2-yl]methyl}dimethylamine
7-(cyclobutylmethyl)-2-[(1-ethyl-1H-pyrazol-5-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
N1-[3-methyl-1-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1,4-dicarboxamide
6-methyl-N-[1-(pyridin-3-yl)pentyl]imidazo[1,2-a]pyridine-2-carboxamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl]propanoic acid
1'-(5-chloro-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-(5-chloropyridine-3-carbonyl)-4-(2-methylquinolin-6-yl)piperidin-4-ol
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(1S)-1-phenylpropyl]pyrimidin-2-amine
4-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}imidazolidin-2-one
N-(1H-1,3-benzodiazol-2-ylmethyl)-6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-{3-[4-(1-hydroxy-2-methylpropyl)piperidine-1-carbonyl]phenyl}propanamide
3-[2-(3,4-difluorophenyl)ethyl]-1-(dimethyl-1,2-oxazole-4-carbonyl)piperidine
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-5-methylpiperidin-2-one
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
(3S,4S)-1-(2-methyl-1H-pyrrole-3-carbonyl)-4-propylpyrrolidine-3-carboxylic acid
6-ethyl-N-[2-(quinolin-8-yloxy)ethyl]pyrimidin-4-amine
1-{[1-(4-amino-5-cyanopyrimidin-2-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
1-[(2-fluoro-3-methoxyphenyl)methyl]-4-[6-(propan-2-yl)pyridin-2-yl]piperazine
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-5-methylimidazo[1,2-a]pyridine-2-carboxamide
1-methyl-2-[4-(6-methylpyridin-2-yl)piperazine-1-carbonyl]azepane
3-[5-(6-phenylpyridazin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]benzonitrile
N-benzyl-2-[4-(4-{[2-(pyrazin-2-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
N-[(2R,3R)-1'-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
2-[(8-methoxy-2H-chromen-3-yl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
2-methyl-6-(propan-2-yl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]pyrimidin-4-amine
1-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-4-(1H-pyrazol-1-yl)butan-1-one
1-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-3-phenylpyrrolidin-3-ol
2-(1,3-thiazol-2-ylmethyl)-4-(3-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}piperidin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
8-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
(3R,5S)-5-(morpholin-4-ylmethyl)-N,1-bis(2-phenylethyl)piperidine-3-carboxamide
N-(1-{7-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-2-(2-oxo-4-phenylpyrrolidin-1-yl)-N-(pyridin-2-ylmethyl)acetamide
(1R,3S)-7-(6-aminopyrimidin-4-yl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1H-pyrazole-4-carboxamide
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-methyl-1H-indole-2-carboxamide
ethyl 2-({2-[benzyl(2-hydroxyethyl)carbamoyl]phenyl}amino)acetate
ethyl 4-(3-phenylpropyl)-1-[2-(pyridin-4-ylsulfanyl)acetyl]piperidine-4-carboxylate
N-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
(1R,5R)-6-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[(2R,3R)-1'-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxybenzamide
3-[2-(2-fluorophenoxy)pyridin-3-yl]-1-[(1-hydroxycyclohexyl)methyl]urea
1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-N-[4-(2-fluorophenoxy)phenyl]piperidine-2-carboxamide
1-[(5-acetylthiophen-3-yl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-[3-(cyclohexylsulfanyl)propyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
2-[(4-fluorophenyl)methyl]-4-(pyridin-4-ylmethyl)morpholine
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)acetamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
8-[(2-chloro-5-fluorophenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-1-(pyridin-4-ylmethyl)pyrrolidin-2-one