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2-amino-4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
1-[(diethylcarbamoyl)methyl]-N-[2-(pyridin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-(cyclopropylmethyl)-8-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-N-[2-(pyrazin-2-yl)ethyl]piperidin-4-amine
4-(3-hydroxy-4-methoxybenzoyl)-5-methyl-1-(2-methylphenyl)piperazin-2-one
2-{4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
N,N-dimethyl-2-[(1S,5R)-3-{[4-(2-methylpropyl)phenyl]methyl}-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-2-(methylsulfanyl)acetamide
(3S,4S)-3-[({4-[(3-fluorophenyl)methoxy]-3-methoxyphenyl}methyl)amino]-4-hydroxy-1λ6-thiolane-1,1-dione
1-{3-[3-(naphthalene-2-carbonyl)piperidin-1-yl]-3-oxopropyl}piperidin-2-one
ethyl 1-(2-{2,5-dioxo-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-yl}acetyl)piperidine-3-carboxylate
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)cyclohex-3-ene-1-carboxamide
4-[2-methyl-7-(1,3-thiazol-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-1,4-oxazepane
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}({[2-(3-methylphenyl)-1,3-thiazol-4-yl]methyl})amine
1-{1-[(1-{furo[3,2-c]pyridin-4-yl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}propan-2-ol
3-(4-methoxy-3,5-dimethylbenzoyl)-N-(2-methoxyphenyl)piperidine-1-carboxamide
2-[6-(1,2,3,4-tetrahydroisoquinolin-5-yl)pyridin-3-yl]acetic acid
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-3-[5-(thiophen-2-yl)furan-2-yl]propan-1-one
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)cyclohexyl]-4-(3-hydroxy-3-methylbutyl)benzamide
2-ethyl-N-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}pyrimidine-5-carboxamide
N-methyl-5-[(3-methyl-2-oxo-1,2-dihydroquinoxalin-1-yl)methyl]-1,2,4-oxadiazole-3-carboxamide
8-[(2S)-2-hydroxy-3-phenylpropanoyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
4-[1-(2,3-difluorobenzoyl)piperidin-3-yl]-2-methyl-5-(3-methylphenyl)pyrimidine
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-6-azaspiro[2.5]octane
2-(3-methoxyphenyl)-1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}ethan-1-one
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperidine
5-(2,4-dimethylbenzoyl)-N-(2-hydroxyethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(3S,4S)-4-cyclopropyl-1-[3-(6-oxo-1,6-dihydropyridazin-3-yl)propanoyl]pyrrolidine-3-carboxylic acid
6-[(3-ethoxy-4-methoxyphenyl)methyl]-N-(2-phenylethyl)-6-azaspiro[2.5]octane-1-carboxamide
methyl 6-[(3,4-dimethylphenyl)methyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-methyl-4-{1-[1-(4-methyl-1H-imidazole-5-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}piperazine
methyl 3-acetamido-1-ethyl-5-{[4-(4-methoxyphenyl)butan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(2-ethoxyethyl)-1-[(3S)-3-hydroxy-3-phenylpropyl]-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
2-(3-chloropyridin-2-yl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
1-(diethylamino)-3-[4-({[2-(4,6-dimethylpyrimidin-2-yl)ethyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
(1S,5R)-6-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
7-[2-amino-6-(2-methylpropyl)pyrimidine-4-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
4-(hydroxymethyl)-1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]piperidin-4-ol
2-(cyclopropylmethyl)-8-(morpholine-4-sulfonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[4-(1H-1,3-benzodiazol-1-yl)phenyl]-3-(dimethylamino)pyrrolidine-1-carboxamide
5-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]pyrrolidin-3-amine
[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl](4-methoxy-4-methylpentan-2-yl)amine
(1-benzofuran-2-ylmethyl)(methyl){[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
1'-[(3-methyl-1,2-oxazol-5-yl)methyl]-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(4aS,8aR)-1-(3-methoxypropyl)-6-(1-methyl-1H-pyrazole-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
5-chloro-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
1-ethyl-8-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-2-oxo-1-phenyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)pyrrolidine-3-carboxamide
2,5-dimethyl-N-(oxan-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine