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1-cyclopropyl-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]({3-methoxy-4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}methyl)amine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)propanamide
1-{1-[2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-methyl-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-N-(2,2,6,6-tetramethylpiperidin-4-yl)propanamide
{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
4-[(E)-2-(furan-2-yl)ethenyl]-3-(thiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(1R,7S)-N-methyl-4-oxo-3-[2-(piperidin-1-yl)ethyl]-N-propyl-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-{4-[(2,2-dimethyloxan-4-yl)methyl]piperazin-1-yl}-6-ethylpyrimidine
4-chloro-1-{2-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethyl}-1H-pyrazole
1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
1-(6-carbamoylpyrazin-2-yl)-4-(2-methylphenoxy)piperidine-4-carboxylic acid
1-[4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-(thiophen-2-yl)ethane-1,2-dione
2-methyl-7-oxo-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
4-(6-methylpyridazin-3-yl)-2-(trifluoromethyl)morpholine
3-[(3S,4R)-1-benzyl-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]-N-[(4-methoxyphenyl)methyl]propanamide
1-(3-chloro-4-methoxyphenyl)-5-oxo-N-[2-(1H-pyrrol-1-yl)ethyl]pyrrolidine-3-carboxamide
2-(2-aminoethyl)-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
4-[(2-aminopyrimidin-5-yl)methyl]-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
2-{5-[6-(methoxymethyl)pyridin-2-yl]-3-methyl-1H-1,2,4-triazol-1-yl}benzoic acid
2-(pyridin-3-yl)-7-(pyridine-3-sulfonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{[5-methyl-2-(2-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}spiro[2.5]octane-1-carboxamide
1-[1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carbonyl]pyrrolidine-2-carboxylic acid
N-tert-butyl-2-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)acetamide
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
11-(benzylamino)-4-[(4-methoxyphenyl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-methyl-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)thieno[2,3-d]pyrimidin-4-amine
N-(4-carbamoyl-2-methylphenyl)-3-(2-methylphenyl)piperidine-1-carboxamide
N-[3-(4-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]furan-2-carboxamide
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[2-(propan-2-yloxy)ethyl]propanamide
1-(2-methoxyethyl)-8-[(4-methoxyphenyl)methyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
{1-[({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]cyclobutyl}methanol
(1S,5R)-3-[(5-methylthiophen-2-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1-[2-(pyrrolidin-1-yl)ethyl]-1,2,3,6-tetrahydropyridine
2-amino-4-(3-chloro-4-hydroxy-5-methoxyphenyl)-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetamide
N-(2-fluoro-4-methylphenyl)-2-{[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]formamido}acetamide
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
1-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-4-phenyl-5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H-imidazole
2-(1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-yl)-6-chloro-1H-1,3-benzodiazole
2-(1-cyclopentyl-4-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperazin-2-yl)ethan-1-ol
(1R,5R)-N,N-dimethyl-6-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]benzamide
[(4-{1-[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-triazin-3-yl]piperidin-2-yl}phenyl)methyl]dimethylamine
3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
N,2-dimethyl-6-propyl-N-[2-(1H-pyrazol-4-yl)ethyl]pyrimidin-4-amine
2-(2,5-dioxoimidazolidin-4-yl)-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)acetamide