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6-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-N-methylpyridine-2-carboxamide
N-[3-(2-methyl-1H-imidazol-4-yl)phenyl]acetamide
6-[(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
N-(1H-1,3-benzodiazol-2-ylmethyl)-2-(cyclopropylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-2-methyl-5-propylpyrimidine
N-[2-(diethylamino)ethyl]-N-methyl-3-(5-methylthiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
N-(2-chloro-4-fluorophenyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carboxamide
5-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-(dimethyl-1,2-oxazol-4-yl)-2-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}acetic acid
N,N-dimethyl-2-{[2-(4-methylpiperazin-1-yl)propanamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N,N,2-trimethyl-7-(3-propyl-1H-pyrazole-5-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl](methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
(1R,3S)-3-(2-hydroxyethoxy)-7-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-7-azaspiro[3.5]nonan-1-ol
1-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-2,4-dimethoxy-N-methylbenzamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-methyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-2-amine
N-[3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N,3,6-trimethyl-1-benzofuran-2-carboxamide
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-phenoxyethan-1-one
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]propanamide
N-[2-(azepan-1-yl)ethyl]-N-methyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
1-cycloheptanecarbonyl-4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]piperidine
(2-{2-[1-(3-fluoropyridine-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
4-(3-methylbutyl)-11-[(propan-2-yl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-methyl-6-[6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-[(3S,4R)-1-(2-methylfuran-3-carbonyl)-4-propylpyrrolidin-3-yl]acetamide
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}propane-1-sulfonamide
2,3,6-trimethyl-N-[1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]quinoline-4-carboxamide
5-acetyl-N-(1-{2-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)thiophene-2-carboxamide
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propan-1-one
N-{[3-(methylsulfanyl)phenyl]methyl}-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
2,6-dimethyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}quinoline-4-carboxamide
N-[1-(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]-2-(thiophen-3-yl)acetamide
N-(1-{7-[(2-chloro-3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
3-phenyl-N-(1-{7-[(2,4,6-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
5-[2-(1H-imidazol-1-yl)acetyl]-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-(2-chloro-4-{[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenoxy)propanoic acid
2-(3-hydroxypropyl)-9-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[2-(4-hydroxypiperidin-1-yl)ethyl]-1-[3-(3-methoxyphenyl)phenyl]urea
(1S,6R)-9-(2-aminopyridine-4-carbonyl)-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
1-[(3-fluorophenyl)methyl]-4-(morpholine-2-carbonyl)-1,4-diazepane
5-(2,6-dimethoxyphenyl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1,2,4-triazin-3-amine
3-(2-oxo-2-{4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}ethyl)-1,3-oxazolidin-2-one
5-{3-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-oxopropyl}imidazolidine-2,4-dione
1-[2-ethoxy-5-(trifluoromethyl)phenyl]-3-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]urea
2-(3-methoxypropyl)-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidine
9-(2,6-dimethylbenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}phenol
N-{[1-(1H-1,3-benzodiazol-2-ylmethyl)pyrrolidin-3-yl]methyl}pyridazine-3-carboxamide