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4-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazole
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-2-(pyridin-2-yl)acetamide
4-(6-chloropyridazin-3-yl)-2-(trifluoromethyl)morpholine
4,6-dimethyl-3-[4-(oxan-4-yl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
2-{3-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
1-(oxolan-2-ylmethyl)-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-(4-{4-phenyl-1-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-imidazol-5-yl}phenyl)ethan-1-one
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]acetamide
1-[2-(furan-2-yl)azepan-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
1-[4-(pyridin-2-yl)pyrimidin-2-yl]piperidine-3-carboxamide
4-[4-(pyrrolidine-1-carbonyl)phenoxy]-1-(thiophen-2-ylmethyl)piperidine
N-(2,5-difluorophenyl)-3-[4-(1,3-thiazol-2-yl)-1H-1,2,3-triazol-1-yl]propanamide
(3R,5S)-N3-(4-fluorophenyl)-N5-(3-methoxypropyl)-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
[4-({1-[1-(pyridine-3-carbonyl)piperidin-4-yl]pyrrolidin-3-yl}methyl)phenyl]methanol
1-[(2-chloro-6-fluorophenyl)methyl]-5-[5-(methoxymethyl)furan-2-yl]-3-methyl-1H-1,2,4-triazole
N-{[5-(dimethylcarbamoyl)furan-2-yl]methyl}-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
3-[2-(dimethylamino)ethyl]-5-[1-(3,4-dimethylbenzoyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
2-cyclopropyl-9-(1H-imidazol-2-ylmethyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
1-{1-[2-(4-methylphenoxymethyl)furan-3-carbonyl]piperidin-3-yl}pyrrolidin-2-one
2-ethyl-N-(2-methoxyethyl)-N-(1,3-thiazol-2-ylmethyl)pyrimidine-5-carboxamide
(4aR,7aS)-1-methyl-4-(4-phenylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}[3-(pyridin-3-yloxy)propyl]amine
2-(2-{[(1-methylpiperidin-4-yl)(2-phenylethyl)amino]methyl}phenoxy)acetamide
(1R,2R,6S,7S)-4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(2,3-dihydro-1-benzofuran-2-ylmethyl)methylamine
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperidin-3-ol
N-[(2-fluorophenyl)methyl]-4-[4-({[3-(1H-pyrazol-1-yl)phenyl]methyl}amino)piperidin-1-yl]benzamide
5-(1-benzyl-1H-pyrazol-3-yl)-4-methyl-N-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1,3-thiazol-2-amine
2-cyclohexyl-N-[(1r,4r)-4-hydroxycyclohexyl]-1,3-benzoxazole-6-carboxamide
4-[(2,3-difluorophenyl)methyl]-3-(2-oxo-2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}ethyl)piperazin-2-one
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-2-(dimethyl-1,2-oxazol-4-yl)-N-[(3S)-2-oxoazepan-3-yl]acetamide
N-[4-(propan-2-yl)phenyl]-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperidin-3-amine
(4aR,7aS)-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N3-[2-(pyridin-2-ylsulfanyl)ethyl]piperidine-1,3-dicarboxamide
2-methoxy-N-{3-methyl-1-[7-(quinolin-6-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}acetamide
N-({1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
N-{[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-1-(propan-2-yl)piperidine-4-carboxamide
(2E)-3-(3-fluorophenyl)-1-{4-[5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}prop-2-en-1-one
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
2-(cyclopropylmethyl)-N-[(4-methylpyridin-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(2R,4R,6S)-2-phenyl-6-[3-(1H-pyrazol-1-ylmethyl)phenyl]oxan-4-yl]acetamide
ethyl 1-(1H-pyrazol-3-ylmethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
2-methoxy-6-({methyl[3-(phenylsulfanyl)propyl]amino}methyl)phenol
2-(cyclohex-1-en-1-yl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]acetamide
4-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
1-[benzyl(methyl)amino]-3-[4-({[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]amino}methyl)phenoxy]propan-2-ol
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-[(3-methylphenyl)methyl]benzamide
4-[({[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]-1-cyclopropylpyrrolidin-2-one
1-[(2E)-3-phenylprop-2-enoyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid