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3-(3,4-difluorophenyl)-5-[2-(1,2-oxazolidin-2-yl)ethyl]-1,2,4-oxadiazole
(1S,5R)-6-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(3-fluorophenyl)-N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}acetamide
N-(2-{7-[(3,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
4-(2-{4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}phenyl)-1λ6-thiomorpholine-1,1-dione
(3S,4S)-1-(4-methoxybenzoyl)-4-[methyl(thiophen-3-ylmethyl)amino]pyrrolidin-3-ol
3-methyl-1-[2-methyl-5-(2-oxopyrrolidin-1-yl)phenyl]-3-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)urea
methyl 5-[(adamantan-2-yl)amino]-3-(2-methoxyacetamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-{[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenol
2-(3-{2-[6-(dimethylamino)pyridin-3-yl]-1H-imidazol-1-yl}phenyl)-N-methylacetamide
3-cyclopentyl-5-[(4-fluorophenyl)methyl]-5-[1-(furan-2-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-3-(4-hydroxyphenyl)benzamide
[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl](methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
(4aS,7aR)-1-(3-methoxypropanoyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-cyclopropyl-N-(2,2-dimethyloxan-4-yl)-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-{[8-(3-phenylpropyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-4-(pyrrolidin-1-yl)benzamide
(3S,4R)-N-(2,3-dihydro-1H-inden-2-yl)-4-ethoxyoxolan-3-amine
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(4-methyl-1,3-thiazol-5-yl)-N-[(1-propyl-1H-pyrazol-4-yl)methyl]propanamide
(1S,5R)-3-(pyridine-4-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[4-oxo-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]benzonitrile
9-methoxy-7-(2-methoxyphenyl)-4-(2-methyl-1,3-thiazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{4-[4-({[4-(trifluoromethyl)phenyl]methyl}amino)piperidin-1-yl]benzoyl}piperidin-3-ol
5-cyclobutyl-N-(oxolan-2-ylmethyl)-1,3,4-oxadiazol-2-amine
3-chloro-N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-4-fluoro-1-benzothiophene-2-carboxamide
N-{1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}methanesulfonamide
{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[(4-phenoxyphenyl)methyl]amine
3-(4-propoxyphenyl)-1,2,4,5,10,11-hexaazatricyclo[7.3.0.02,6]dodeca-3,5,7,9,11-pentaene
(2S,4R)-4-(4-{2-[(3-chlorophenyl)formamido]propan-2-yl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
5-[1-(4-fluorophenyl)cyclopropyl]-3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazole
(3S,4R)-4-(hydroxymethyl)-1-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}piperidin-3-ol
2-methyl-7-[3-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl 6-(2-cyclohexylacetyl)-2-[(2-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}pyrimidine-5-carboxamide
3-benzoyl-N-(1-hydroxybutan-2-yl)-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
1-(4-methoxy-2-{[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenyl)-1H-pyrazole
4-{2-[2-(cyclopropylmethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-3-(1H-indol-3-yl)propan-1-one
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-methyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
(2E)-1-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}-3-(thiophen-2-yl)prop-2-en-1-one
7-fluoro-N,2-dimethyl-N-[(5-methylthiophen-2-yl)methyl]quinoline-4-carboxamide
methyl 9-(cyclopentyloxy)-3-(3-methylbut-2-en-1-yl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[(4-chlorophenyl)methyl]-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-1,3-benzoxazole-5-carboxamide
3-{2-[2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]-4-methylphenyl}-1,3-oxazolidin-2-one
N-[(3R,4S)-1-(3-hydroxypropyl)-4-propylpyrrolidin-3-yl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-{1-[2-(1H-pyrazol-1-yl)benzoyl]piperidin-3-yl}benzoic acid
2-{[5-methoxy-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-yl]amino}-N-methylethane-1-sulfonamide
2-(2-chloro-4-fluorophenoxymethyl)-N-[2-(1H-pyrazol-1-yl)ethyl]-1,3-oxazole-4-carboxamide
1-[2-(dimethylamino)-6-(5-methyl-1,3-oxazole-4-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-ol
3-(3-ethylphenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid