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5-[1-(3-methylpentanoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
4-(3-cyanopiperidine-1-carbonyl)-N-(2,2-difluoroethyl)benzene-1-sulfonamide
1-[2-(methylamino)acetyl]-4-(oxan-4-yl)-1,4-diazepane-6-carboxylic acid
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-[2-(1H-imidazol-1-yl)acetyl]-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-2-carboxamide
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)[4-(morpholin-4-yl)butyl]amine
4-({8-[(5-methylpyrazin-2-yl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)benzonitrile
2-({2-[5-(oxan-2-yl)thiophen-2-yl]-1H-imidazol-1-yl}methyl)pyridine
2-(1-cyclohexyl-4-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-3-(4H-1,2,4-triazol-4-yl)benzamide
3-acetamido-N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}propanamide
(1S,5R)-3-[2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)acetyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
5-{3-[2-(methoxymethyl)piperidin-1-yl]-3-oxopropyl}-5-(naphthalen-1-ylmethyl)pyrrolidin-2-one
3-(2,5-dichlorophenyl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
7-[(3-phenoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1-cyclopropyl-4-[({[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]pyrrolidin-2-one
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[3-(furan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
4-[(3Z)-hex-3-en-1-yl]-1-[(2R)-pyrrolidin-2-ylmethyl]-1H-1,2,3-triazole
3-[4-(5-aminopyridin-3-yl)-3,5-dimethyl-1H-pyrazol-1-yl]propanamide
4-{4-[2-(trifluoromethyl)pyrimidin-4-yl]piperazine-1-carbonyl}morpholine
N-[(2,4-difluorophenyl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]pyrazine
methyl 6-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}pyrimidine-4-carboxylate
2-cyclopropyl-8-[2-(ethylamino)pyrimidine-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
1-[(3-methoxyphenyl)methyl]piperidin-3-amine
3-(5-methylthiophen-2-yl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
methyl 3-(2,3-dihydro-1,4-benzodioxine-6-sulfonamido)-5-[(2,2-dimethylpropanamido)methyl]benzoate
(1S,5R)-3-(3-chloro-4-fluorobenzoyl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}-2-(2-ethyl-1H-imidazol-1-yl)ethan-1-one
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl){[4-(methylsulfanyl)phenyl]methyl}amine
N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)prop-2-ene-1-sulfonamide
9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-3-(4,4,4-trifluorobutyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-7-methyl-3H,4H-thieno[3,2-d]pyrimidin-4-one
[4-(1-benzoxepine-4-carbonyl)-1,4-oxazepan-6-yl]methanol
N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-2-(1H-pyrrol-1-yl)propanamide
N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-2-(trifluoromethyl)benzamide
5-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-(oxolan-2-ylmethyl)-4-[4-(quinolin-4-ylmethyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
2-cyclopentyl-9-(4-hydroxybenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(1-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
2-[1-(5-ethyl-1,2-oxazole-3-carbonyl)-4-(pyrrolidin-1-ylmethyl)piperidin-4-yl]-5-methylpyridine
1-({5-[(4-butoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
1-{1-[(2-butyl-1H-imidazol-4-yl)methyl]azepan-4-yl}-3-phenylurea
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]acetamide
4-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]pyridine
6-fluoro-3-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-3,4-dihydroquinazolin-4-one
N-[(4-acetamidophenyl)methyl]-2-{[(2-methylpyridin-4-yl)methyl]amino}acetamide