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(5-{1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
5-(2-methoxyacetamido)-1-methyl-2-(pyridin-4-yl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
3-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[2-(morpholin-4-ylmethyl)phenyl]urea
N-{[1-(3-ethyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]methyl}acetamide
N-[(1S,2R,4R)-bicyclo[2.2.1]heptan-2-yl]-5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazole-3-carboxamide
6-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-N,N-dimethylpyridine-3-carboxamide
{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(trifluoromethyl)phenyl]methyl}amine
2-({6-[2-(4-chlorophenyl)morpholin-4-yl]pyrimidin-4-yl}amino)ethan-1-ol
N-[4-({[(2,3,5-trimethyl-1H-indol-7-yl)methyl]amino}methyl)phenyl]acetamide
N-cyclopentyl-3-methyl-N-[(5-methylthiophen-2-yl)methyl]-4-oxo-3,4-dihydroquinazoline-7-carboxamide
(2S,4R)-4-amino-N-methyl-1-[2-(methylsulfanyl)benzoyl]pyrrolidine-2-carboxamide
1-(2-methoxy-4-{[methyl(prop-2-en-1-yl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
(2S)-1-(3-cyclopentaneamidobenzoyl)pyrrolidine-2-carboxylic acid
2-ethoxy-3-{[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl}pyridine
1-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}-4-(thiophen-2-ylmethyl)piperazine
methyl 2-[5-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)-1H-pyrazol-3-yl]acetate
N-[3-hydroxy-1-(4-methylphenyl)propyl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
7-methyl-2-[3-(2-oxoimidazolidin-1-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
1-{1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carbonyl}azetidin-3-ol
4-(diethylamino)-N-methyl-N-[1-(pyridin-3-yl)ethyl]benzamide
2-(2-methylpropyl)-8-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
1-(2,3-dihydro-1H-indol-1-yl)-2-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]ethane-1,2-dione
(3R,4R)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
4-[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]-5-methanesulfonyl-2-methylpyrimidine
(2S,4R)-4-butanamido-N,N-diethyl-1-(4-methylpyrimidine-5-carbonyl)pyrrolidine-2-carboxamide
5-chloro-3-(1,2-oxazol-3-ylmethyl)-3,4-dihydroquinazolin-4-one
6-{2-[(2-chlorophenyl)methyl]morpholine-4-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-N-[(5-methylpyrazin-2-yl)methyl]pyrimidin-2-amine
1-[3-(4-fluorophenoxy)propyl]-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperazine
ethyl 4-(2-methoxyethyl)-1-[3-(morpholin-4-yl)propanoyl]piperidine-4-carboxylate
N-[(2-chlorophenyl)methyl]-N-methyl-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
1-(3-chlorophenyl)-4-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-5-methylpiperazin-2-one
2-{2-[2-(methylsulfanyl)phenyl]-1H-imidazol-1-yl}acetamide
N-methyl-3-(4-methylthiophen-2-yl)-N-[2-(pyridin-2-yl)ethyl]-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
4-(1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)pyrimidine
3-{6-oxa-9-azaspiro[4.5]decan-9-ylmethyl}benzoic acid
1-(2,3-dihydro-1H-inden-2-yl)-4-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]-1,4-diazepane
3-(1-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carbonyl}piperidin-2-yl)pyridine
1-(2-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-2,7-diazaspiro[4.5]decan-7-yl)ethan-1-one
5-[(E)-2-(4-hydroxy-3-methoxyphenyl)ethenyl]-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
3-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-4-methylbenzene-1-sulfonamide
5-[(1S,5R)-6-(2-methoxyethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid
methyl 4-{[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}benzoate
methyl 3-{[(1-methylpiperidin-3-yl)methyl](2-phenylethyl)carbamoyl}propanoate
6-{[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-2-cyclopropylpyrimidin-4-ol
3-methyl-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pentanamide
benzyl[(4-methyl-1,3-thiazol-5-yl)methyl](oxolan-3-ylmethyl)amine
(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)[(1-methyl-1H-indol-3-yl)methyl]amine
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[2-(methylamino)-1,3-thiazole-4-carbonyl]piperidin-4-ol
4-{1-phenyl-4-[1-(pyridin-4-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrazol-3-yl}pyridine