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methyl 4-{4-[1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazin-1-yl}benzoate
[3-(2-phenylethyl)-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-3-yl]methanol
(1-{[1-(2-chloro-4,5-difluorobenzoyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
3-tert-butyl-1-[(1-propylpiperidin-4-yl)methyl]urea
N-[(4-methyl-1H-imidazol-2-yl)methyl]-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)cyclopentanamine
2-(1H-imidazol-2-yl)-N-[(5-methylpyrazin-2-yl)methyl]benzamide
ethyl 4-{6-oxo-3-phenyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}-1H-pyrazole-3-carboxylate
(1S,6R)-9-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
3-methoxy-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
5-(2-fluorophenoxymethyl)-3-[3-(2-methylpropyl)pyrrolidine-1-carbonyl]-1H-pyrazole
4-[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]-2-[(1-hydroxycyclohexyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-{1-cyclopentyl-7-[2-(methoxymethyl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl}benzamide
N-ethyl-4-({[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl}amino)piperidine-1-carboxamide
1-methyl-4-{3-[2-(methylsulfanyl)ethyl]-5-(pyrrolidin-3-yl)-1H-1,2,4-triazol-1-yl}-1,2-dihydroquinolin-2-one
propyl 3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
methyl[(3-{[1-(naphthalene-2-sulfonyl)piperidin-4-yl]oxy}phenyl)methyl](thiophen-3-ylmethyl)amine
1-[4-(adamantan-1-yl)piperazin-1-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
1-(4-ethylpiperazin-1-yl)-3-[1-(3-fluoro-4-methoxybenzoyl)piperidin-4-yl]propan-1-one
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-3-(1-methyl-1H-pyrazol-5-yl)propanamide
2-[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]-1H-1,3-benzodiazole-5-carboxylic acid
methyl 1-benzyl-5-[(2,2-dimethylpropyl)amino]-3-(oxolane-2-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(2-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-2-yl}ethyl)phenol
2-{5-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
{1-[3-(isoquinolin-1-yl)phenyl]ethyl}dimethylamine
2-(2,4-difluorophenyl)-5-(furan-3-ylmethyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepine
1-({4-[(3-methoxyphenyl)carbamoyl]phenyl}methyl)-N-methylpyrrolidine-3-carboxamide
ethyl 1-{4-[(2-methylpyridin-3-yl)oxy]piperidine-4-amido}cyclobutane-1-carboxylate
2-cyclopropyl-9-[2-(methylsulfanyl)acetyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-(dimethylamino)-7-[2-(1H-1,2,4-triazol-3-yl)benzoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-(oxolan-2-ylmethoxy)acetamide
N-(1-{3-[3-(methoxymethyl)piperidine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)-2-(3-methylphenyl)acetamide
(3S,4R)-4-phenyl-1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]pyrrolidine-3-carboxylic acid
N4-[2-(2,4-dimethoxyphenyl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
(2-{2-[1-(2-ethylpyrimidine-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methylfuran-2-carboxamide
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]oxane-4-carboxamide
7-(3,6-dimethylpyrazin-2-yl)-4-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{1-[3-(2-methoxyphenyl)propanoyl]piperidin-3-yl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
4-methyl-1-[7-(oxolan-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-1,4-diazepan-5-one
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
2-[1-(1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]propan-2-ol
7-{[4-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
4-[(3-aminoazepan-1-yl)methyl]-5-tert-butylfuran-2-carboxamide
(1S,5R)-3-(5-phenylpentanoyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(1-benzofuran-2-ylmethyl)-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
2-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]-N-ethyl-N-methylpyrimidin-4-amine
4-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]-7-{[4-(pyridin-2-ylmethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}-4-(2-methoxyphenoxy)piperidine
(2S,4R)-1-benzyl-4-{[(4-fluorophenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide