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1-[2-(dimethylamino)-4-{[3-(2-ethyl-1H-imidazol-1-yl)propyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)urea
(1R,3s,6r,8S)-4-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-azatricyclo[4.3.1.13,8]undecane
(1-{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)methanol
2-(dimethylamino)-2-(3-methylphenyl)-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
(1S,5R)-3-cyclobutanecarbonyl-6-(2-methoxypyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-methylbut-2-en-1-one
(2R,3R,6R)-5-(5-fluoro-2-methylbenzoyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[3-(cyclohexyloxy)propyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
1-[(4-ethyl-1,3-thiazol-2-yl)methyl]-4-(5-ethylfuran-2-yl)-1H-1,2,3-triazole
N-(7-{6-azabicyclo[3.2.1]octane-6-carbonyl}-1-methyl-2-phenyl-1H-1,3-benzodiazol-5-yl)ethane-1-sulfonamide
1-phenyl-4-({[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}amino)pyrrolidin-2-one
2-methyl-3-[3-(1H-pyrazol-3-yl)phenyl]pyrazine
N-[(3,4-difluorophenyl)methyl]-3-[1-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)piperidin-3-yl]propanamide
1-(5-ethylpyrimidin-2-yl)-4-(pyridin-3-ylmethyl)-1,4-diazepane
4-hydroxy-N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-1-methylpiperidine-4-carboxamide
N-[(3R,4R)-3-hydroxy-1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]pyridine-2-carboxamide
3-[(4-fluorophenyl)methyl]-N-[2-(propan-2-yloxy)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
[(3S,5R)-1-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}-5-[(dimethylamino)methyl]piperidin-3-yl]methanol
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-cyclopentylpyrimidine
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{[1-(dimethylamino)cyclohexyl]methyl}-1H-pyrazole-3-carboxamide
(3R,4R)-3-cyclobutyl-1-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-4-methylpyrrolidin-3-ol
2,3,5-trimethyl-N-[2-(pyridin-3-yloxy)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
methyl 3-cyclobutaneamido-5-[(oxan-4-yl)amino]-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
9-(1,2,4-oxadiazol-3-ylmethyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-2-[(quinolin-6-yloxy)methyl]-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
1-[2-({[1-(hydroxymethyl)cyclopentyl]methyl}(methyl)amino)pyrimidin-4-yl]piperidin-3-ol
methyl (2S)-2-{[5-(2-methoxyacetamido)-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazol-7-yl]formamido}-2-phenylacetate
{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}[(5-ethylpyridin-2-yl)methyl]methylamine
2-amino-6-(4-hydroxy-2-methylphenyl)-4-[4-(2-hydroxyethoxy)phenyl]pyridine-3-carbonitrile
3-[(2-{1-[(1R,2S,3S,4R,5S)-tricyclo[3.2.1.02,4]octane-3-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)methyl]pyridine
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-[2-(4-chlorophenyl)ethyl]-N-methyl-N-[2-(oxan-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
2-(2-butyl-1H-imidazol-4-yl)-1-(2,2,2-trifluoroethyl)-1H-imidazole
N-ethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
(2S)-2-({[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)-4-methylpentanamide
4-oxo-5-phenoxy-1-[1-(1H-pyrazol-1-yl)propan-2-yl]-1,4-dihydropyridine-3-carboxylic acid
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-5-(1H-imidazol-1-ylmethyl)-N-methylpyridin-2-amine
2-(2H-indazol-2-yl)-1-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
3-(4-methyl-1,3-thiazol-5-yl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}propanamide
3-cyclopentaneamido-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-4-methylbenzamide
N-{2-[(3-{[(4-hydroxy-3-methoxyphenyl)methyl]amino}-5-[(2-methylphenyl)sulfamoyl]phenyl)formamido]ethyl}acetamide
(4aS,8aR)-6-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridine-4a-carboxylic acid
2-[(4-chlorophenyl)methyl]-N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1,3-benzoxazole-5-carboxamide
4-{4-methyl-6H,7H,8H-cyclopenta[g]quinolin-2-yl}piperazin-2-one
N-(2-tert-butyl-6-methylphenyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
(2S)-3-methyl-2-{4-[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]-1H-1,2,3-triazol-1-yl}butanamide
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-methyl-3-(1H-1,2,4-triazol-1-yl)propan-1-one
8-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2-methyl-2,8-diazaspiro[4.5]decane