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(4aR,8aR)-2-cyclopentanecarbonyl-7-(3-phenylpropyl)-decahydro-2,7-naphthyridin-4a-ol
3-fluoro-N-(1-hydroxybutan-2-yl)-8-methyl-N-(thiophen-2-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
5-[(2-chlorophenyl)methyl]-3-(cyclopropylmethyl)-5-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
N-[2-(furan-2-yl)ethyl]-2-methyl-7-(piperidin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-5-(2-methylpropyl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-(2-methoxyphenyl)-N-methyl-N-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]-1H-pyrazole-4-carboxamide
2,5-dimethyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
methyl (1R,3S,3aR,6aS)-1-ethyl-5-methyl-3-(naphthalen-2-yl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
2-methyl-4-(4-methylphenyl)-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazine
1-(3-{2,8-diazaspiro[4.5]decan-2-ylmethyl}phenyl)ethan-1-one
(1R,3R,5S)-8-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-hydroxy-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(4-methylphenyl)pyrimidine-5-carboxamide
4-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-ylmethyl]-N-methyl-1,3-thiazol-2-amine
3-ethyl-5-(2-{2-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1H-imidazol-1-yl}ethyl)-1,2,4-oxadiazole
3-[5-(oxolan-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
7-[(1-ethyl-1H-imidazol-5-yl)methyl]-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(1-methoxy-2-methylpropan-2-yl)piperidine-3-carboxamide
6-ethyl-1,5-dimethyl-3-[2-(trifluoromethyl)morpholine-4-carbonyl]-1,2-dihydropyridin-2-one
1-(2-methylpyridin-4-yl)-4-[2-(methylsulfanyl)benzoyl]-1,4-diazepane
(5-{[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}furan-2-yl)methanol
{1-[(2-ethoxyphenyl)methyl]-4-[(4-methoxyphenyl)methyl]piperidin-4-yl}methanol
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(2-hydroxyphenyl)methyl]-N-methylacetamide
(2S)-2-{[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-4-(methylsulfanyl)butan-1-ol
N-methyl-N-(oxan-4-yl)-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(3-methoxybenzoyl)piperazine
N5-[2-(diethylamino)ethyl]-N6-(3-methoxypropyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
methyl 3-(7-chloro-2-{[(4-acetamidophenyl)formamido]methyl}-2,3-dihydro-1-benzofuran-5-yl)benzoate
propyl 4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-{1-[(5-ethylfuran-2-yl)methyl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
N-methyl-N-[(5-methylfuran-2-yl)methyl]-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methanesulfonyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}acetamide
7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N,N-diethyl-1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazole-5-carboxamide
3-{2-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-1,2,3-thiadiazole-4-carboxamide
(3R)-1-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]pyrrolidin-3-ol
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
4-[(4-methyl-5-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
2-methyl-5-{[4-(3,3,4-trimethylpiperazine-1-carbonyl)-1,3-oxazol-2-yl]methoxy}-1,3-benzothiazole
methyl 5-{[(2-chloro-6-fluorophenyl)methyl]amino}-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(3S,5R)-1-(2-cyclopentylacetyl)-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
N-(2-fluoroethyl)-1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-amine
(1S,5R)-6-(1-methyl-1H-indole-2-carbonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-[(3,4,5-trimethoxyphenyl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-phenyl-7-{[4-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine