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5-({[1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)-1,3,4-thiadiazol-2-amine
N-(2-methoxyethyl)-3-(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)propanamide
N-tert-butyl-2-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}acetamide
5-amino-3-[1-(4-methylpyridin-2-yl)-1H-pyrrol-2-yl]-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
2-{1-[(2-fluorophenyl)methyl]-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazin-2-yl}ethan-1-ol
4-acetyl-N-(1,4-oxazepan-6-ylmethyl)-3,4-dihydro-2H-1,4-benzoxazine-6-sulfonamide
2-(3-methoxypropyl)-8-(6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-(4-methoxyphenyl)-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
1-[(3-fluorophenyl)methyl]-4-(pyrazine-2-carbonyl)piperazin-2-one
(4aS,8aS)-4a-hydroxy-N-{4-[(2-methoxyethyl)carbamoyl]phenyl}-decahydroisoquinoline-2-carboxamide
5,5-dimethyl-3-(2-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidine-2,4-dione
1-(furan-3-carbonyl)-4-(3-methylphenoxy)piperidine
5-(2-methyl-1H-imidazol-4-yl)-1-(2-methylprop-2-en-1-yl)-4-phenyl-1H-imidazole
methyl 2-{[2-(2,6-dimethoxyphenoxy)ethyl](methyl)amino}acetate
N-{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-4-fluoro-N-(oxolan-2-ylmethyl)benzamide
1-cycloheptyl-N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
3-[(4-{1-[(3-fluoro-2-methylphenyl)methyl]pyrrolidin-3-yl}piperidin-1-yl)methyl]pyridine
N-(2H-1,3-benzodioxol-5-yl)-1-(1,2-oxazol-3-ylmethyl)piperidin-3-amine
4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-(4-methoxy-3,5-dimethylphenyl)piperidine-1-carboxamide
{1-[2-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]piperidin-2-yl}methanol
1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-4-(trimethyl-1H-pyrazole-4-carbonyl)-1,4-diazepane
3-(2-fluorophenyl)-6-(furan-2-ylmethyl)-1-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-[2-(1H-imidazol-4-yl)ethyl]-9-[(5-methylthiophen-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[5-(2-methanesulfonamidoethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]acetic acid
2-[4-({4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
[(3R,4R)-1-{[4-(cyclopentyloxy)phenyl]methyl}-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
4-(4-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-imidazol-2-yl}phenyl)but-3-yn-1-ol
N-{[8-(2-phenylpropyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}furan-2-carboxamide
1-(2-methylhexanoyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(3S,4R)-1-[2-methyl-2-(morpholin-4-yl)propyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
(4aS,7aR)-1-[(5-chlorothiophen-2-yl)methyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl({[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}){[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-{5-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1,2,4-oxadiazol-3-yl}pyridine
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}[(5-methylthiophen-2-yl)methyl]amine
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-[(furan-2-ylmethyl)amino]pyridine-3-carboxamide
2-[({1-[(3,4-difluorophenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)amino]-N-methylacetamide
1-(2,4-dimethylphenoxy)-3-({2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)propan-2-ol
1-(cyclohex-3-en-1-ylmethyl)-3-(4-ethyl-1H-pyrazol-5-yl)piperidine
4-(4-methylphenoxy)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-ethoxy-5-methylbenzene-1-sulfonamide
(5S)-5-({[(8-fluoro-4-hydroxyquinolin-2-yl)methyl](pyridin-2-ylmethyl)amino}methyl)pyrrolidin-2-one
2-methyl-N-[3-(morpholin-4-yl)propyl]-4-oxo-1,4-dihydroquinoline-8-carboxamide
8-(4-chlorobenzoyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2,2-dimethylpropan-1-one
(3aR,6aR)-2-(1-benzylpiperidin-4-yl)-5-(2-hydroxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[2,4-bis(trifluoromethyl)benzoyl]-1,4-oxazepan-6-ol
4-{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperidin-4-yl}thiomorpholine
2-{9-[3-(2-methylphenyl)propanoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
1-[4-(2-methoxy-5-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenoxy)piperidin-1-yl]ethan-1-one
N-[(2-chlorophenyl)methyl]-N-(2-hydroxyethyl)-3-methoxy-2,2-dimethylpropanamide