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N-(2H-1,3-benzodioxol-5-yl)-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperidin-3-amine
2-(4-methoxyphenyl)-N-({1-[(1-methyl-1H-indol-3-yl)methyl]piperidin-3-yl}methyl)acetamide
12-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-15-methyl-9-(pyridin-2-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one
4-[(5-fluoro-2-methylphenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}furan-3-carboxamide
5-(2,6-difluorophenoxymethyl)-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[1-(pyrazin-2-yl)propan-2-yl]-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazolin-2-amine
7-fluoro-N,2-dimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}quinoline-4-carboxamide
methyl 4-(4-{2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetyl}piperazin-1-yl)benzoate
N-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-1H-pyrazole-4-carboxamide
2-methyl-3-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraene
5-{1-[3-(4-methylphenyl)propanoyl]piperidin-4-yl}-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-{2-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
(3R,4R)-4-cyclopropyl-1-[(5-fluoro-2-methoxyphenyl)methyl]-3-methylpiperidin-4-ol
2-{1-[(5-methylfuran-2-yl)methyl]-4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
2-{5-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]-1H-pyrazol-3-yl}pyridine
9-methoxy-N-methyl-7-oxo-N-(1,3-thiazol-4-ylmethyl)-3-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-{[3-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]methyl}-5,5-dimethylimidazolidine-2,4-dione
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[3-(pyrazin-2-yl)propanoyl]piperidine-2-carboxamide
2-methoxy-N-(1-{7-[(4-methoxy-2,3-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)acetamide
1-(4-aminopyrimidin-2-yl)-4-[1-(methoxymethyl)cyclopropanecarbonyl]-1,4-diazepan-6-ol
2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1-[1-(2-fluorobenzoyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-(butan-2-yl)-6-chloro-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
4,6-dimethyl-3-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-1,2-dihydropyridin-2-one
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3-fluorophenyl)acetamide
N-[3-(dimethylamino)propyl]-1-(4-fluorobenzenesulfonyl)-N-methylpiperidin-3-amine
4-[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
4-[1-(2-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]-1-phenylpiperazin-2-one
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-4-(2-oxopiperidin-1-yl)butanamide
2-[4-(2-oxo-6-phenyl-1,2-dihydropyridine-3-carbonyl)morpholin-3-yl]acetic acid
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[4-(4-methoxypyrimidin-2-yl)piperazin-1-yl]propan-1-one
3-(2-cyclohexylacetyl)-N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[2-(2-methylpiperidine-1-carbonyl)phenyl]acetamide
2-[4-(2,6-diaminopyrimidin-4-yl)-1-[(4-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
4-(1-acetylpiperidine-4-carbonyl)-6-methyl-1-[2-(methylsulfanyl)phenyl]piperazin-2-one
1-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)-3-methoxypiperidine
(2E)-N-{[2-(4-acetylpiperazin-1-yl)-6-methylquinolin-3-yl]methyl}-N-[2-(cyclohex-1-en-1-yl)ethyl]-3-(3-fluorophenyl)prop-2-enamide
2-{3-[2-(3-fluorophenyl)ethyl]piperidine-1-carbonyl}pyrazine
N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-6-{[(1r,4r)-4-hydroxycyclohexyl]amino}pyridine-3-carboxamide
7-(4-ethylbenzenesulfonyl)-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-[2-(1H-imidazol-1-yl)ethyl]-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidine
2-{[2-(methoxymethyl)piperidin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
methyl 3-(2-cyclopentylacetyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
dimethyl({1-[1-(2-methylpentyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)amine
N-[(2S)-1-[4-benzyl-3-oxo-6-(pyridin-3-ylmethoxy)-1,4-diazepan-1-yl]-4-(methylsulfanyl)-1-oxobutan-2-yl]acetamide
4-[3-(methanesulfonylmethyl)piperidin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
1-(2-benzyl-1,3-thiazole-4-carbonyl)-2-(1-methyl-1H-pyrazol-3-yl)piperidine
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-1,2,3-thiadiazole-4-carboxamide
3-({2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}[(5-methylthiophen-2-yl)methyl]amino)propan-1-ol