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2-[1-methyl-10-oxo-4-(thiophen-3-ylmethyl)-1,4,9-triazaspiro[5.6]dodecan-9-yl]acetic acid
1-(2-{[methyl(propyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)-2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethan-1-one
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
N,1-dimethyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl 2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-1-methyl-1H-1,3-benzodiazole-5-carboxylate
2-{1-ethyl-5-[(pyridin-2-ylsulfanyl)methyl]-1H-1,2,4-triazol-3-yl}acetamide
2-(3-phenylpropyl)-4-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]morpholine
5-{2-[3-(oxolan-3-yl)-1-propyl-1H-1,2,4-triazol-5-yl]phenyl}-1H-1,2,3,4-tetrazole
(2R)-2-amino-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-2-phenylacetamide
N3-cycloheptyl-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
methyl 1-[(3S,5S)-5-{[2-(1H-indol-3-yl)ethyl]carbamoyl}-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-[(3-methoxyphenyl)methyl]-2-(6-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(prop-2-en-1-yl)acetamide
3-{1-[(2-ethylpyrimidin-4-yl)methyl]piperidin-4-yl}propanamide
2-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}ethan-1-ol
5-(dimethylamino)-2-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2,3-dihydropyridazin-3-one
{[2-chloro-5-ethoxy-4-(propan-2-yloxy)phenyl]methyl}(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)amine
1-benzyl-N3-methyl-4-oxo-N3-(2-phenylethyl)-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-(4-ethoxyphenyl)-3-(1H-1,2,3,4-tetrazol-5-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[(4-methoxy-3-methylphenyl)methyl]-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazin-2-one
4-(benzylamino)-1-(6-hydroxy-4-methyl-1,4-diazepan-1-yl)butan-1-one
1-(cyclopropylmethyl)-4-(1H-imidazol-2-ylmethyl)-2-(propan-2-yl)-1,4-diazepane
N-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
4-(1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)benzoic acid
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-{[(3-phenoxyphenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
(2S,3S)-3-methyl-2-[(2-methyl-1-benzofuran-7-yl)formamido]pentanamide
4-{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}morpholine
2-(4-chloro-2-methylphenoxy)-N-(1H-imidazol-2-ylmethyl)-N-methylacetamide
2-{3-[1-(4-chlorophenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}acetamide
(2H-1,3-benzodioxol-5-ylmethyl)(methyl)[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-[2-(2-phenylethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
4-(2,3-dihydro-1H-isoindole-2-carbonyl)-1-[2-(dimethylamino)ethyl]pyrrolidin-2-one
3-(4-chloro-1H-pyrazol-1-yl)-1-[(3S,4S)-3-hydroxy-4-(thiomorpholin-4-yl)pyrrolidin-1-yl]propan-1-one
2-(methylamino)-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}pyridine-4-carboxamide
(1S,5R)-6-propyl-3-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{2-[4-(3-fluorophenoxy)piperidin-1-yl]-2-oxoethyl}-3-(2-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
N-[4-({[(3S)-2-oxoazepan-3-yl]carbamoyl}methoxy)phenyl]propanamide
N-[(3R,4R)-1-[(4-cyano-5-methyl-1H-pyrrol-2-yl)methyl]-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
N-{2-[(1E)-pent-1-en-1-yl]pyridin-3-yl}cyclopropanecarboxamide
4-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-1-(2-methoxyphenyl)-2,2-dimethylpiperazine
N-propyl-5-[5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazol-2-yl]pyrimidin-2-amine
3-ethyl-N-(quinolin-5-yl)-1,2-oxazole-5-carboxamide
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)[(3-methylthiophen-2-yl)methyl]amine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-N-methyl-6-oxopiperidine-3-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-1-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-{4-[2-amino-3-cyano-6-(2-methylpropanoyl)-5,6,7,8-tetrahydro-1,6-naphthyridin-4-yl]phenyl}acetamide
(1S,5R)-3-[5-(methoxymethyl)furan-2-carbonyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[4-(2-aminopyridine-4-carbonyl)-1-(3-phenylpropyl)piperazin-2-yl]ethan-1-ol
(3R,5S)-N-butyl-5-(morpholin-4-ylmethyl)-1-(2-phenylethyl)piperidine-3-carboxamide
4-methyl-6-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-2-amine
8-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one