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1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
5-(3-phenylpropyl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
4-[(3-fluorophenyl)methyl]-3-[2-(morpholin-4-yl)-2-oxoethyl]piperazin-2-one
5-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
4-chloro-2-{[methyl(quinolin-2-ylmethyl)amino]methyl}phenol
(4aR,7aS)-1-propanoyl-4-(5-propylthiophene-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-benzyl-3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]piperazin-2-one
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
N-{[7-(3,5-difluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
methyl 3-[2-(3-methoxyphenyl)acetyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(thiophen-2-ylmethyl)piperazine
5-chloro-6-oxo-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1,6-dihydropyridine-3-carboxamide
3-{[(1H-1,3-benzodiazol-2-ylmethyl)(methyl)amino]methyl}-1-(cyclohexylmethyl)-3-hydroxypiperidin-2-one
2-(dimethylamino)-2-(3-fluorophenyl)-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
1-(1-benzofuran-2-ylmethyl)-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-{3,9-diazaspiro[5.5]undecan-3-yl}-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
{[3-({1-[4-(3-fluorophenyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}(furan-3-ylmethyl)methylamine
3-ethyl-8-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[3-(4-methoxyphenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(thiophen-2-ylmethyl)acetamide
8-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-methylphenyl)methyl]acetamide
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]pyridine-3-carboxamide
(4S,4aS,8aR)-1-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-phenyl-decahydroquinolin-4-ol
2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-(quinolin-6-ylmethyl)acetamide
4-methoxy-4-(prop-2-en-1-yl)-N-(quinolin-6-yl)piperidine-1-carboxamide
5-[1-(3,5-difluorobenzoyl)piperidin-4-yl]-3-[2-(dimethylamino)ethyl]-5-(2-phenylethyl)imidazolidine-2,4-dione
9-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(1H-imidazol-2-yl)benzoyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
4-[6-(propan-2-yl)-2-(trifluoromethyl)pyrimidin-4-yl]piperazine-2-carboxylic acid
({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)(quinolin-2-ylmethyl)amine
4-(1H-indole-5-carbonyl)-7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{4-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidine-1-carbonyl]phenyl}ethan-1-one
N-[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]-3-(1,2-oxazinan-2-yl)propanamide
N-{1-[(3-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
1-[4-(piperidin-3-ylmethyl)benzoyl]-4-(pyridin-4-yl)-1,4-diazepane
2,3-dimethyl-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
2-(2-ethoxyphenyl)-2-[4-(piperidine-1-carbonyl)piperidin-1-yl]acetic acid
1-{3-[(2-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-4-methylpentane-1,2-dione
1-ethyl-N-[2-(3-methoxyphenyl)ethyl]-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(3-methoxypropyl)-8-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
1-[(4-cyanophenyl)methyl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-{5-[2-(4-fluorophenyl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
methyl (2R)-2-(4-hydroxyphenyl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridin-3-ylformamido}acetate
1-[2-hydroxy-3-(2-methoxy-4-{[(naphthalen-1-ylmethyl)amino]methyl}phenoxy)propyl]piperidin-4-ol
N-[2-(2-fluorophenyl)ethyl]-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}-N-methyloxolan-3-amine
1-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4,4,4-trifluorobutan-1-one
2-methyl-N-[({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}carbamoyl)methyl]propanamide
(1R,3S)-3-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}cyclopentan-1-amine