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N-{2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}adamantane-1-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}cyclopent-1-ene-1-carboxamide
1-(4-methoxybutyl)-4-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperazine
{1-[(2,5-difluorophenyl)methyl]-4-(3-phenylpropyl)piperidin-4-yl}methanol
3-[1-(1-cyclopropyl-5-oxopyrrolidine-3-carbonyl)piperidin-4-yl]-N-(2,3-dihydro-1,4-benzodioxin-6-yl)propanamide
(1R,7S)-N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-4-oxo-3-(pentan-3-yl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-methyl-N-(pyrimidin-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-3-methyl-1H-pyrazole-5-carboxamide
N-[(2-methoxyphenyl)methyl]-N-[(3-methylphenyl)methyl]pent-4-ynamide
N-[3-(3-ethylphenoxy)propyl]-N-methyl-1-(pyrimidin-2-yl)piperidine-4-carboxamide
N-(furan-2-ylmethyl)-7-(3-methoxypropanamido)-N,1-dimethyl-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
5-(3-acetylphenoxymethyl)-N-[(2R)-1-hydroxy-3-methylbutan-2-yl]-1H-pyrazole-3-carboxamide
methyl 3-({[4-(3-fluorophenyl)phenyl]formamido}methyl)-5-(pyridine-4-amido)benzoate
(4aS,7aR)-1-({2-[2-(dimethylamino)ethoxy]phenyl}methyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-(2-methoxyethyl)-2-(5-methoxyfuran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-[2-(methylsulfanyl)ethyl]-3-phenyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-ethoxy-6-[1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenol
8-(oxolan-3-yl)-3-{3-[4-(propan-2-yl)piperazin-1-yl]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(3ar,6ar)-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-4-[(6-chloropyridin-3-yl)methyl]piperazine
2-{2-[4-(6-methoxypyridin-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1,2,3,4-tetrahydrophthalazine-1,4-dione
7-{[(butan-2-yl)(pyridin-3-ylmethyl)amino]methyl}-4-methyl-2H-chromen-2-one
4-{[7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]methyl}benzoic acid
(3S,4S)-4-cyclopropyl-1-[1-(4-methoxyphenyl)piperidin-4-yl]pyrrolidine-3-carboxylic acid
3-(cyclopropylmethyl)-5-[2-(4H-1,2,4-triazol-4-yl)phenoxymethyl]-1,2,4-oxadiazole
N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
(4aS,7aR)-1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4aR,7aS)-1-cyclopropanecarbonyl-4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-benzyl-4-{[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl}piperazine
1-(5-ethyl-2-methylpyrimidin-4-yl)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-amine
(2R,3S)-2-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-hydroxybutanamide
2-(2-aminoethyl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]quinazolin-4-amine
3-(3-fluorophenyl)-N-[1-(pyrazin-2-yl)piperidin-4-yl]-1H-pyrazole-4-carboxamide
1-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}-3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}propan-1-one
1-[2-(3-fluorophenyl)ethyl]-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-6-oxopiperidine-3-carboxamide
(1R,3S)-3-({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}(methyl)carbamoyl)cyclopentane-1-carboxylic acid
6-chloro-N,N-dimethyl-3-{[(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)amino]methyl}imidazo[1,2-a]pyridine-2-carboxamide
5-[2-(2-methyl-1H-indol-3-yl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N'-(2-chlorophenyl)-N-(prop-2-en-1-yl)-N-(propan-2-yl)ethanediamide
4-(2-chloro-3,4-dimethoxyphenyl)-1-(1-methylpiperidin-4-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(3S)-2-oxoazepan-3-yl]-3-(1H-pyrazol-1-ylmethyl)-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}benzamide
2-{[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}benzonitrile
6-(propan-2-yl)-N4-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidine-2,4-diamine
2-(2-fluorophenyl)-1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
5-amino-4-chloro-N-[(4-phenyloxan-4-yl)methyl]-1H-pyrazole-3-carboxamide
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
5-(3-phenylpropyl)-5-{1-[(2,3,4-trimethoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
N-(4-{[4-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}phenyl)acetamide
1-(2,6-difluoro-4-methoxybenzoyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
N-[4-(pyridin-3-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]oxolane-3-carboxamide
N-(1-methyl-1H-1,3-benzodiazol-6-yl)-3-(2-methylpiperidin-1-yl)azetidine-1-carboxamide