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3-{5-[(5-cyclopentylthiophen-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-dimethylpiperazine-1-carboxamide
9-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H,2H,3H,6H,7H,8H,9H-[1,4]oxazino[3,2-g]quinoline-2,7-dione
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-{[(1-phenylcyclopropyl)amino]methyl}piperidin-2-one
1-{2-[2-(4-fluorophenyl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
[(3R,4R)-1-(4-ethyl-5-methylthiophene-3-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
5-[3-(2-ethoxyethoxy)phenyl]-1-methyl-1H-1,2,4-triazole
1-[(4-fluoro-3-methoxyphenyl)methyl]piperidine-3-carbonitrile
N-{[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(1H-pyrazol-3-yl)benzamide
N3-methyl-N5-[(4-methylphenyl)methyl]-N3-(2-methylpropyl)-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
6-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-N,N-dimethylpyrimidin-4-amine
1-(piperidin-1-yl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]cyclohexane-1-carboxamide
3-[(5-methyl-1H-imidazol-4-yl)methyl]-5-(piperidin-4-yl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1-(propan-2-yl)piperidine-4-carboxamide
4-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-3-ethylmorpholine
3-methyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1-[2-(morpholin-4-ylmethyl)phenyl]urea
5-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-1,2-dihydropyridin-2-one
2-(3,5-difluorophenyl)-N-(1H-imidazol-2-ylmethyl)-N-methylacetamide
(4aR,8aS)-1-[2-(3,4-dimethoxyphenyl)ethyl]-6-(furan-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-[2-(dimethylamino)ethyl]-3-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methylbenzamide
2-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido
3-(1,4-diazepane-1-sulfonyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
N-[1-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
1-[(1-methyl-1H-pyrazol-5-yl)methyl]-2-[2-(thiophen-2-yl)ethyl]piperidine
3-(1-methyl-1H-pyrazol-4-yl)-N-[2-(propane-2-sulfonyl)ethyl]propanamide
4,4,4-trifluoro-1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]butan-1-one
2-(2H-1,3-benzodioxol-5-yl)-1-{9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}ethan-1-one
(1-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}piperidin-4-yl)methanamine
2-[2-(dimethylamino)ethyl]-9-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
(2S)-N-methyl-5-oxo-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]pyrrolidine-2-carboxamide
ethyl 3-(2-methoxyethyl)-1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-3-carboxylate
3-[(4aR,7aS)-4-[(4-acetylphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
7-(2-hydroxyethyl)-2-[3-(6-oxo-1,6-dihydropyridazin-3-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-3-carboxamide
3,5-dihydroxy-4-methyl-N-{[1-(oxan-4-yl)pyrrolidin-3-yl]methyl}benzamide
N-[(3S,4R)-4-(4-methylphenyl)-1-[2-(pyridin-3-yl)acetyl]pyrrolidin-3-yl]acetamide
4-[1-(2-phenylethyl)-5-(pyridine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
2-methylpropyl 9-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-3,9-diazaspiro[5.5]undecane-3-carboxylate
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
4-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1-cyclopropylpyrrolidin-2-one
5-[3-cyclopropyl-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1-methyl-1H-pyrrole-3-carbonitrile
4-(4-chlorophenoxy)-N-[2-(1H-imidazol-1-yl)ethyl]piperidine-4-carboxamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
N-[2-(3-{[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}phenoxy)propyl]-4-(2-oxopyrrolidin-1-yl)benzamide
2-(benzyloxy)-1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
(3R,4S)-4-cyclopropyl-1-[3-(pyridin-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-amine
3-(3-acetylphenyl)-6-[(3-acetylphenyl)methyl]-1-methyl-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
5-(naphthalen-1-yl)-3-[4-(pyrrolidin-1-yl)piperidin-1-yl]-1,2,4-triazine
1-(2-chlorophenyl)-4-[2-(pyridin-3-yl)-1H-imidazol-1-yl]pyrrolidin-2-one
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine