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({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl){[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}amine
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
4-hydroxy-N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-1-methylpiperidine-4-carboxamide
methyl 3-{[2-(2-{4-[(propan-2-yl)carbamoyl]-1H-1,2,3-triazol-1-yl}ethyl)piperidin-1-yl]sulfonyl}thiophene-2-carboxylate
2-(3-methyl-1H-pyrazol-5-yl)-6-(pyrrolidine-1-carbonyl)pyrazine
1-cyclohexyl-4-(3-phenoxypropanoyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
(1-{[1-(1,3-benzothiazol-2-ylmethyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
1-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
[(2-methoxyphenyl)methyl][(6-methylpyridin-2-yl)methyl](prop-2-en-1-yl)amine
2-[5-oxo-3-(3,3,3-trifluoropropyl)-4,5-dihydro-1H-1,2,4-triazol-4-yl]propanoic acid
1-[2-(3-hydroxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-2-phenylethane-1,2-dione
1-[(5-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-4-methylpiperazine
1-(cyclopropylmethyl)-3-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-(1-methylpiperidin-4-yl)pyridin-2-amine
(2S,4R)-4-amino-1-(cyclopropanesulfonyl)-N-ethylpyrrolidine-2-carboxamide
3-methyl-3-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-[4-(trifluoromethoxy)phenyl]urea
(3S,4R)-1-[2-(methylamino)acetyl]-4-phenylpyrrolidine-3-carboxylic acid
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2,4-dimethylpyrimidine-5-carboxamide
2-(2-chloro-4-{[4-(hydroxymethyl)-4-methylpiperidin-1-yl]methyl}phenoxy)propanoic acid
1-{3-[(4-cyclopentylpyrimidin-2-yl)amino]propyl}piperidin-4-ol
3-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}propan-1-one
1-{2-[5-(1,4-dimethylpiperidin-4-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyrrolidin-2-one
2-(3-methylbutyl)-8-(1,3-thiazol-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-butyl-8-[2-(2-methyl-1H-indol-3-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-3-(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)propanamide
3-({3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
5-chloro-3-methyl-N-[(5-methylpyrazin-2-yl)methyl]-1H-indole-2-carboxamide
1-[2-({ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-6-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
4-{[3-(2-fluorophenoxy)azetidin-1-yl]methyl}-1-(propan-2-yl)-1H-pyrazole
N-[(2,3-dimethylphenyl)methyl]-5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
1-(2-{1-[(3,4-dimethoxyphenyl)methyl]piperidin-2-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
7-[(3-methylphenyl)methyl]-2-(2-methylpyridine-3-carbonyl)-2,7-diazaspiro[4.5]decane
(4S)-3-[(2-methoxypyridin-3-yl)methyl]-4-(propan-2-yl)-1,3-oxazolidin-2-one
1-[(2S,4R)-1-[(2,5-dimethoxyphenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carbonyl]-4-(1-methylpiperidin-4-yl)piperazine
1-cyclobutanecarbonyl-N-(3,4-dimethylphenyl)piperidin-3-amine
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-2-(thiophen-3-yl)acetamide
naphthalen-1-yl (7S,9aR)-7-[(4-chlorophenyl)methyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
1-(2,3-dihydro-1-benzofuran-2-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-cyclohexyl-4-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-4-(3-methylpyridin-4-yl)-1,4-diazepane
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-(thiophen-3-yl)-1H-pyrazole-5-carboxamide
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
5-ethyl-N,2,3-trimethyl-N-[2-(pyrrolidin-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-{2-[({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amino]ethyl}piperidin-3-ol
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(pyrrolidin-1-yl)propan-1-one
1-{7-[(5-butylthiophen-2-yl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}ethan-1-one
8-[(2-chlorophenyl)carbamoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(2,3-dihydro-1H-inden-1-yl)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)acetamide
1-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole