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3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}propanamide
methyl 3-[(2E)-3-(4-fluorophenyl)prop-2-enamido]-6-{[2-(2-hydroxyethyl)piperidin-1-yl]methyl}thieno[2,3-b]pyridine-2-carboxylate
1-[(3-methoxyphenyl)methyl]-6-oxo-N-[2-(pyridin-4-yl)ethyl]piperidine-3-carboxamide
2-chloro-4-({[2-(1H-imidazol-4-yl)ethyl]carbamoyl}amino)-N-propylbenzamide
N-ethyl-1-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
(1S,3R)-3-amino-N-[(4-methoxyphenyl)methyl]-N-(pyridin-4-ylmethyl)cyclopentane-1-carboxamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
1-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
2-[4-cyclohexyl-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
4-[4-(1H-imidazol-1-ylmethyl)phenyl]-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-[2-({2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
N-[2-(ethylsulfanyl)ethyl]-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-cyclobutanecarbonyl-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]piperidine-4-carboxamide
(1S,6R)-3-methyl-9-{2-methylpyrido[2,3-d]pyrimidin-4-yl}-3,9-diazabicyclo[4.2.1]nonan-4-one
N-{2-[(2-fluoro-5-sulfamoylphenyl)formamido]ethyl}pyridine-3-carboxamide
4-[7-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
(3aS,6aR)-5-(3,6-dimethylpyrazin-2-yl)-3-[2-(4-methoxyphenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-cyclopentyl-N'-[2-hydroxy-3-(3-methoxyphenoxy)propyl]butanediamide
6-[3-(benzyloxy)piperidin-1-yl]-N-(2-methoxyethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
ethyl 5-{[(furan-2-ylmethyl)amino]methyl}-1-(4-phenyl-1,3-thiazol-2-yl)-1H-pyrazole-4-carboxylate
5-[1-(furan-3-carbonyl)pyrrolidin-2-yl]-N-methyl-N-(1H-pyrazol-5-ylmethyl)thiophene-2-carboxamide
2-{[1-(2-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1-ethyl-1H-imidazole
2-({1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-3-yl}methyl)-1H-1,3-benzodiazole
3-(4-cyclopentylphenyl)-6-methylpyridazine
1-(cyclopropylmethyl)-N-methyl-5-(3-phenoxypropanoyl)-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(4-fluorophenoxymethyl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1,3-oxazole-4-carboxamide
5-methyl-4-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-N-(pyrimidin-4-ylmethyl)benzene-1-sulfonamide
ethyl 2-[methyl({1-[4-(5-phenylpentanamido)phenyl]piperidin-4-yl})amino]acetate
5-(3-ethyl-1H-indole-2-carbonyl)-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-4-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
1-(furan-2-ylmethyl)-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]piperidine-4-carboxamide
2-(dimethylamino)-2-(3-methylphenyl)-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]acetamide
N-(2,3-dihydro-1H-inden-5-yl)-2-{4-[(2-methyl-1,3-oxazol-4-yl)methyl]morpholin-3-yl}acetamide
(2S)-2-(2-{[(2-chlorophenyl)methyl]sulfanyl}acetamido)propanamide
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetamide
4-chloro-N,1-dimethyl-N-(1-methylpyrrolidin-3-yl)-1H-pyrazole-3-carboxamide
N-[3-(2-methyl-1H-imidazol-1-yl)propyl]-9H-purin-6-amine
2-(4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
1,5-dimethyl-4-{[(1R,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-pyrrole-2-carbonitrile
N-{[4-methoxy-3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-[1-(3-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-1-methylpiperidine
(3R,4S)-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-4-propylpyrrolidin-3-amine
5-methyl-2-(2-methylphenyl)-4-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1,3-oxazole
1-methoxy-3-[(2-methylquinolin-4-yl)amino]propan-2-ol
dimethyl({[(1R,5S,6S)-3-({2-phenylimidazo[1,2-a]pyridin-3-yl}methyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine
1-[(2,5-dimethylphenyl)methyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
1-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
1-(1H-1,3-benzodiazole-5-carbonyl)-4-(2-phenoxyethyl)piperidine-4-carboxylic acid
2,4-dimethyl-N-(2-{7-[(2-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide