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2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1,3-oxazole-4-carboxamide
N-{2-[2-(1-phenylethyl)-1H-imidazol-1-yl]ethyl}acetamide
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[(2-methylphenyl)methyl]benzamide
1-(4-chlorophenyl)-N-[(3S,4S)-4-methoxy-1,1-dioxo-1λ6-thiolan-3-yl]cyclobutane-1-carboxamide
N-cyclopentyl-3-[5-(1,3-thiazol-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
(2S,4S)-N-ethyl-1-[(4-methyl-1H-imidazol-2-yl)methyl]-4-[3-(methylsulfanyl)propanamido]pyrrolidine-2-carboxamide
6-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octane
1-[3-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-3-oxopropyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(2-fluorophenyl)methyl]-4-[1-(propan-2-yl)piperidine-4-carbonyl]-1,4-diazepane
3-(pentan-2-yl)-1-{4-[2-(pyridin-2-yl)ethoxy]phenyl}urea
4-(1-ethyl-1H-imidazol-2-yl)-1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]piperidine
8-(2-fluorobenzoyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
N-tert-butyl-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl][1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
N,N-dimethyl-2-{[2-(pyridin-4-ylsulfanyl)acetamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-ethyl-6-methyl-2-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-1,2-dihydropyridine-4-carboxamide
N-{[(3S,4S)-3-hydroxy-1-[2-methyl-2-(morpholin-4-yl)propyl]piperidin-4-yl]methyl}pyrrolidine-1-carboxamide
methyl 2-(cyclopentylsulfamoyl)-6-(2,3-dimethylbenzoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-(1-{7-[(4-phenylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxane-4-carboxamide
N-(2-hydroxyethyl)-N-[(2-methylphenyl)methyl]-4-sulfamoylbenzamide
2,6-dimethyl-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]pyrimidine-4-carboxamide
1-cyclopentyl-N3-methyl-N3-(2-methylpropyl)-4-oxo-N5-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
4-[2-amino-3-cyano-6-(1H-indol-3-yl)pyridin-4-yl]benzamide
3-(3-hydroxy-3-methylbutyl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}benzamide
[(1-{[1-(1H-indole-5-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]dimethylamine
2-(cyclopropylmethyl)-9-(4-methoxy-3-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-3-{1-[3-(2-fluorophenyl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}propanamide
3-(5-{[2-(1-phenylethyl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyridine
N-(2-ethoxypropyl)-3-{methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]sulfamoyl}benzamide
2-hydroxy-N-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-carboxamide
1-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-[2-(methylsulfanyl)propyl]-1H-1,2,3-triazole
6-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrazine-2-carboxamide
3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3,4-dihydroquinazolin-4-one
(4S,4aS,8aS)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-phenyl-decahydroquinolin-4-ol
5-hydroxy-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]pyrazine-2-carboxamide
4-{[7-chloro-4-(morpholin-4-yl)quinazolin-2-yl]methyl}-1-phenylpiperazin-2-one
5-{1-[(2,4-dimethoxyphenyl)methyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
ethyl 4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carboxylate
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
3-{4-oxo-4-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]butyl}-3,4-dihydroquinazolin-4-one
(2S,4S)-1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-ethyl-4-(2-methoxyacetamido)pyrrolidine-2-carboxamide
1-(4-{6-[(propan-2-yl)amino]pyridazin-3-yl}phenyl)ethan-1-one
4-[(2-methylphenyl)methyl]-1-[4-(1H-pyrazol-1-yl)benzoyl]-1,4-diazepan-5-one
2-[(2,2-dimethyloxan-4-yl)(ethyl)amino]-N-[(4-acetamidophenyl)methyl]acetamide
1-(4-{[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}thiophen-2-yl)ethan-1-one
4-ethyl-3-{1-[3-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}propanamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(1H-imidazol-2-yl)benzoyl]piperidin-3-ol
2-amino-4-(3-ethenylphenyl)-6-(2-hydroxypropan-2-yl)pyridine-3-carbonitrile
2-(furan-2-yl)-N-(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)-2-oxo-N-(prop-2-en-1-yl)acetamide