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N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
4-{4-[(2-chloro-6-fluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-methylpiperidin-4-ol
6-methyl-5-[5-(1H-pyrazol-3-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
5-fluoro-N-[2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-1H-indole-2-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-cyclohexyl-5-[(5-methyl-1H-pyrazol-1-yl)methyl]-3-(oxan-4-yl)-1H-1,2,4-triazole
N-({3-methyl-7-[4-(trifluoromethyl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)methanesulfonamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carboxamide
3-(2,8-dimethylquinoline-3-carbonyl)-3,9-diazaspiro[5.6]dodecan-10-one
methyl 3-(2-methoxybenzamido)-5-{[2-(thiophen-3-yl)acetamido]methyl}benzoate
4-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4H-1,2,4-triazole
2-chloro-4-{[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidin-1-yl]methyl}-6-methoxyphenol
4-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-6-methylpyrimidin-2-amine
methyl 2-{2,7-diazaspiro[4.5]decane-2-sulfonyl}benzoate
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-2-(pyridin-2-yl)acetamide
2-hydroxy-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-2-phenylethan-1-one
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]acetamide
N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
2-methyl-3-[(4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}piperidin-4-yl)oxy]pyridine
N-(1H-imidazol-2-ylmethyl)-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
[4-(6-ethyl-2-methylquinoline-4-carbonyl)-1,4-oxazepan-6-yl]methanol
8-(2,3-dihydro-1H-inden-2-yl)-3-[2-(dimethylamino)ethyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(3-methanesulfonamidophenyl)-4-(pyridin-4-yl)piperidine-1-carboxamide
2-cyclopentyl-9-(3-hydroxy-4-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(5-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}thiophen-3-yl)prop-2-yn-1-ol
6-methyl-4-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
2-[5-(2-cyclopropylpyrimidin-5-yl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)-5-{1-[2-(1,3-thiazol-4-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
2-(4-{5-[(dimethylamino)methyl]furan-2-carbonyl}-1-(furan-3-ylmethyl)piperazin-2-yl)ethan-1-ol
[(3R,4R)-1-(2-phenylbenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-(carbamoylmethyl)-2-[1-(2-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
3-methyl-2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine
2-({4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylpyridazine-4-carboxamide
N-(2-methoxyethyl)-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)-N-(thiophen-3-ylmethyl)propanamide
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-3-pentanamidobenzamide
(3S,4S)-4-[4-(4-methoxybenzenesulfonyl)piperazin-1-yl]-1-methylpyrrolidin-3-ol
5-{1-[(2,6-difluorophenyl)methyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(2-ethyl-6-methylpyrimidin-4-yl)piperidin-3-ol
{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(ethyl)(pyridin-4-ylmethyl)amine
3-amino-1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]pyrrolidine-3-carboxylic acid
3-(3-fluorophenyl)-4-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)piperazin-2-one
1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-2-(2-phenylethyl)piperidine
2-{[(4-fluorophenyl)methyl](methyl)amino}-1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]ethan-1-one
7-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
5-{[1-(oxan-4-yl)pyrrolidin-3-yl]methyl}-1,2-dihydropyridin-2-one
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
4-(1-benzyl-1H-imidazol-2-yl)-1-(2,6-difluorobenzoyl)piperidine
methyl 3-[(2,6-difluorophenyl)methyl]-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate