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2-amino-6-(1-benzofuran-2-yl)-4-(1H-imidazol-4-yl)pyridine-3-carbonitrile
(1S,5R)-6-(2-methoxyethyl)-3-(4-methyl-1H-imidazole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{3,5-dimethyl-4-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]-1H-pyrrol-2-yl}ethan-1-one
(3R,4R)-1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-ol
4-{[2-(2-fluorophenoxy)ethyl]amino}-2-methylpentan-2-ol
4-{[1-(1-{thieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methyl}piperazin-2-one
N-[(5-chlorothiophen-2-yl)methyl]-3-[(3-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-N-(pyridin-3-ylmethyl)cyclopropanamine
(3S,4R)-1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
(1S,3R)-N-[(3,4-difluorophenyl)methyl]-3-[2-(1H-imidazol-1-yl)acetamido]cyclopentane-1-carboxamide
1-{2-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-[1-(thiophen-2-yl)ethyl]piperidine-3-carboxamide
1-[4-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,3-benzodiazole
4-(4-phenyl-1H-pyrazol-5-yl)-1-(thiophene-2-carbonyl)piperidine
1-[(2-fluorophenyl)methyl]-N-[(1-phenylcyclopentyl)methyl]-1H-1,2,3-triazole-4-carboxamide
(1R,5R)-6-(2-methoxyethyl)-3-(5-methyl-4-phenylthiophene-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-(4-methyl-1H-imidazole-2-carbonyl)-7-{[3-(pyridine-3-carbonyl)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
N-[(2R,3R)-2-methoxy-1'-(1-phenylcyclopropanecarbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
2-[5-(3-acetylphenyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]acetic acid
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[3-(pyridin-3-yl)propyl]benzamide
ethyl 3-(3-phenylpropyl)-1-[3-(pyridin-4-yl)propanoyl]piperidine-3-carboxylate
2-[1'-(oxane-4-carbonyl)-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl]acetamide
3-[ethyl(2,2,2-trifluoroethyl)sulfamoyl]-N-(pyrrolidin-3-yl)benzamide
methyl 5-{[(2,5-dimethylphenyl)methyl]amino}-1-ethyl-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N6-cyclopropyl-N4-methyl-N4-(oxan-2-ylmethyl)pyrimidine-2,4,6-triamine
2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
methyl({[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}){[1-(2-methylpropyl)piperidin-4-yl]methyl}amine
(2S,4R)-N-(1-benzothiophen-2-ylmethyl)-1-[(2-chlorophenyl)methyl]-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-N-methylpyrrolidine-2-carboxamide
4-(5-chloro-2-ethoxyphenyl)-2,5,6-trimethylpyrimidine
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]ethane-1-sulfonamide
methyl 3-[6-methoxy-3-oxo-4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]propanoate
(2R,4S)-4-hydroxy-1-[3-(2-methoxyphenyl)propanoyl]piperidine-2-carboxylic acid
1-(4-methoxyphenyl)-5-methyl-4-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperazin-2-one
1-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]-4-phenylpiperazine
1-[2-methoxy-1-(pyridin-2-yl)ethyl]-1-methyl-3-[1-(propan-2-yl)-1H-pyrazol-5-yl]urea
1-(2,3-dimethoxybenzoyl)-2-(4-fluorophenyl)azetidine
1-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
1-{4-[1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-yl]-1,4-diazepan-1-yl}ethan-1-one
2,5-dimethyl-N-(2-oxoazepan-3-yl)-1,3-thiazole-4-carboxamide
2-[4-({4-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)piperazin-1-yl]pyrimidine
2-(aminomethyl)-N-[4-(3-methoxyphenoxy)phenyl]piperidine-1-carboxamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(methylamino)ethan-1-one
N-ethyl-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(pyridin-4-yl)piperidin-4-yl]oxy}benzamide
N-[(3R,4S)-4-cyclopropyl-1-(2-methanesulfonylethyl)pyrrolidin-3-yl]-3-(1H-pyrazol-1-yl)propanamide
N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-2,3-dihydro-1-benzofuran-7-carboxamide
methyl 2-(4-{4-ethyl-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2,5-dioxoimidazolidin-4-yl}piperidine-1-carbonyl)benzoate
methyl 1-{3-[(3,5-difluorophenyl)methyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperidine-2-carboxylate
N-[1-(4-fluorophenyl)-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]-1H-pyrazole-3-carboxamide
4-[(3-methylphenyl)sulfanyl]-1-[5-(oxolan-2-yl)thiophene-2-carbonyl]piperidine