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N-[(5-methylpyrazin-2-yl)methyl]-3-(pyridin-4-yl)propanamide
N4-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
N-[2-(oxan-2-yl)ethyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
N-({7-[(3-ethoxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2,6-difluorobenzamide
2-[(4aR,7aS)-4-(3-methoxypropanoyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
3,5-dimethyl-1-[1-(2-methyl-1-benzofuran-5-carbonyl)azetidin-3-yl]-1H-pyrazole
(3aS,6aS)-2-(ethanesulfonyl)-5-(3-methoxybenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-chloro-1-({3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}methyl)-1H-pyrazole
5-(pyrrolidine-1-carbonyl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyridin-2-amine
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(1,2-oxazole-3-carbonyl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
methyl (2S,4S)-4-(4-fluorobenzamido)-1-[(3-fluorophenyl)methyl]pyrrolidine-2-carboxylate
(2S,4R)-4-(3-fluorobenzamido)-N-[2-(1H-indol-3-yl)ethyl]pyrrolidine-2-carboxamide
1-{2-hydroxy-3-[3-(morpholin-4-ylmethyl)phenoxy]propyl}piperidin-4-ol
1-(3,3-diphenylpiperidin-1-yl)-2-hydroxypropan-1-one
4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-1-(3-methylphenyl)-1H-pyrazole
3-({[(1-ethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
6-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-N-[2-(2-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
4-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-1-methyl-2-phenylpiperazine
N-methyl-1-[3-(1H-pyrazol-1-yl)phenyl]-N-(pyrimidin-4-ylmethyl)piperidin-4-amine
6-[3-fluoro-5-(trifluoromethyl)phenyl]-N-methylpyridine-2-carboxamide
1-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]-2-(4-methoxyphenoxy)ethan-1-one
(4aS,7aR)-1-(3,5-dimethylbenzoyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
N-cyclopropyl-2-(6-hydroxy-4-{[5-(hydroxymethyl)furan-2-yl]methyl}-1,4-diazepan-1-yl)acetamide
N-methyl-N-(1,2-oxazol-3-ylmethyl)-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-2-(3,4-dimethoxyphenyl)-N-methylacetamide
N-[(3,4-dimethoxyphenyl)methyl]-4-(4-fluorophenyl)-N-(pyridin-2-ylmethyl)benzamide
6-(2-fluoro-4-methoxyphenyl)-7-methyl-2-(4-methyl-1,4-diazepane-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
methyl 4-({3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamido}methyl)benzoate
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
3-chloro-N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-fluoro-N-methylbenzamide
5-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
ethyl 1-methanesulfonyl-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
3-[5-(2,6-dimethylpyrimidin-4-yl)-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-(2-fluorobenzenesulfonyl)-N-methylpiperidin-3-amine
5-(4-benzylpiperidine-1-carbonyl)-N-(furan-2-ylmethyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(4-fluorophenyl)-4-(2-methyl-6-propylpyrimidin-4-yl)piperazine-2-carboxamide
(isoquinolin-5-ylmethyl)(methyl){[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}amine
(4aS,7aR)-1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-1-[4-(morpholin-4-ylmethyl)phenyl]urea
4-cyclobutaneamido-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]benzamide
N-ethyl-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
N-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-2-(3-methoxyphenyl)pyrrolidine-1-carboxamide
(1R,3S)-3-(2-hydroxyethoxy)-7-{[4-(1H-imidazol-1-yl)phenyl]methyl}-7-azaspiro[3.5]nonan-1-ol
2-{[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]methyl}-4-methoxyphenol
2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}-N-[2-(pyridin-3-yl)ethyl]acetamide
6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
N-{2-[(pyridin-3-yl)amino]ethyl}-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
1-ethyl-5-methyl-N-[1-(thiophene-2-carbonyl)piperidin-3-yl]-1H-pyrazole-4-carboxamide