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2,7,8-trimethyl-N-[3-(4H-1,2,4-triazol-4-yl)propyl]quinoline-4-carboxamide
2-{[4-(2,2-dimethylpropyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-6-ethoxyphenol
(1S,5R)-3-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3,9-diazabicyclo[3.3.2]decan-10-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[3-(1H-imidazol-1-yl)propyl]piperidine-3-carboxamide
2-{2-[(dimethylamino)methyl]phenoxy}pyridine-3-carboxamide
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-(2,2-diphenylethyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}acetamide
1-ethyl-4-{1-[2-(oxan-2-ylmethoxy)ethyl]piperidin-4-yl}piperazine
(3R,5S)-N-[3-(dimethylamino)propyl]-5-(3-fluorophenoxymethyl)-1-(2-methylpropyl)piperidine-3-carboxamide
6-(2-fluoro-3-methoxyphenyl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
4-[(1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methyl]morpholine
2-(2-{4-phenyl-5-[6-(trifluoromethyl)pyridin-3-yl]-1H-imidazol-1-yl}ethyl)pyrazine
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(3S,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]propan-1-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-1-(propan-2-yl)piperidine-4-carboxamide
8-(1,3-benzothiazole-5-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{1-[(4-ethoxyphenyl)methyl]-4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
3-(2-chlorophenyl)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}propanamide
5-(2,4-difluorophenoxymethyl)-N-[2-(pyridin-3-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[2-(1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)ethyl]acetamide
(2-methoxyethyl)[(4-methylphenyl)methyl](pyridin-2-ylmethyl)amine
1-[4-({[2-(4-chlorophenyl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
1-cycloheptyl-N-[2-(pyridin-3-yloxy)propyl]-1H-1,2,3-triazole-4-carboxamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]acetamide
4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-N-(1-methylpiperidin-3-yl)pyrimidin-2-amine
methyl 5-{[(3,5-dimethylphenyl)methyl]amino}-3-(2-methoxyacetamido)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(4aR,7aS)-1-(2-methoxyethyl)-4-[3-(2-oxopyrrolidin-1-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)propyl]-1H-1,2,3-benzotriazole
1-[(4aR,8aR)-4a-hydroxy-7-{[4-(2-methylpropyl)phenyl]methyl}-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-[(3R,4S)-1-cyclopentyl-4-cyclopropylpyrrolidin-3-yl]-3-(methylsulfanyl)propanamide
5-chloro-4-{[7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}-2-methoxyphenol
4-(2-{2-[2-(thiophen-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}ethyl)morpholine
1-[(4-fluorophenyl)methanesulfonyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-1,3-oxazole-4-carboxamide
N-[2-(dimethylamino)ethyl]-5-(6-oxopiperidine-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(2S,4S)-4-amino-N,N-diethyl-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]pyrrolidine-2-carboxamide
2-methoxy-5-{[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]methyl}benzoic acid
(2S,4R)-4-amino-1-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]-N-methylpyrrolidine-2-carboxamide
4-(4-methoxyphenoxy)-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine
6-fluoro-2-oxo-N-(oxolan-2-ylmethyl)-N-propyl-1,2-dihydroquinoline-4-carboxamide
1-{3-[3-(benzyloxy)piperidin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
3-[5-({2-[5-(oxolan-2-yl)thiophen-2-yl]-1H-imidazol-1-yl}methyl)-1,2,4-oxadiazol-3-yl]pyridine
4-[3-methyl-5-(phenoxymethyl)furan-2-carbonyl]-2-(trifluoromethyl)morpholine
(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-(2-phenoxyethyl)piperidin-4-yl)methanol
1-cyclopentanecarbonyl-N-[1-(4-hydroxyphenyl)propyl]piperidine-4-carboxamide
5-ethyl-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
3-[(3R,4S)-4-(dimethylamino)-1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl]propanoic acid
3-{[4-({[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}amino)-6-methylpyrimidin-2-yl]amino}phenol
(2R)-1-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-phenylpropan-1-one
4-{[4-(furan-2-yl)phenyl]methyl}-2-(2-methoxyethyl)morpholine