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(2,1,3-benzoxadiazol-5-ylmethyl)({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
4-methyl-2-{2-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
2-({4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}methyl)pyridine
(1-{[methyl({[(1s,4s)-4-aminocyclohexyl]methyl})amino]methyl}cyclopentyl)methanol
methyl 4-(5-{[methyl(oxolan-3-yl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
(1S,6R)-9-(pyridin-2-ylmethyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
N,N-dimethyl-1-[2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidin-4-amine
3-{2-[4-(dimethyl-1,3-thiazol-4-yl)phenyl]ethyl}-1λ6-thiolane-1,1-dione
1-methyl-5-{4-phenyl-5-[2-(prop-2-en-1-yloxy)phenyl]-1H-imidazol-1-yl}piperidin-2-one
2-[4-(1-benzofuran-2-ylmethyl)-1-(2-phenylethyl)piperazin-2-yl]ethan-1-ol
(2R,3R,6R)-5-benzoyl-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-methyl-N-{[7-(quinolin-4-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}butanamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-(2-methoxyphenyl)acetamide
N-(2-hydroxy-2-phenylethyl)-N-(pyridin-4-ylmethyl)imidazo[1,2-a]pyrimidine-2-carboxamide
N-[2-(2-methoxyphenyl)ethyl]-6-{[2-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
2-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
4-methyl-2-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-3,4-dihydro-2H-1,4-benzoxazine
N-{3-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-oxopropyl}methanesulfonamide
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methylpyrrolidine-3-carboxamide
4-{[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine
methyl 4-(4-{2-[3-(2-methoxyphenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]acetyl}piperazin-1-yl)benzoate
2-cyclopropyl-8-[3-(ethylsulfanyl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[1-(2,5-difluorophenyl)cyclopropyl]-1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)urea
1-{7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-4,4,4-trifluorobutan-1-one
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-6-(dimethylamino)pyridine-3-carboxamide
{1-[1-(3-methoxypyrazin-2-yl)piperidin-4-yl]ethyl}dimethylamine
9-(cyclopropylmethyl)-1-methyl-4-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
1-cyclobutanecarbonyl-N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]piperidine-4-carboxamide
(3R)-3-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidine-1-carbonyl}-1,2,3,4-tetrahydroisoquinoline
4-(furan-2-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
1-(4-{[5-(3-chloro-4-methylphenyl)furan-2-yl]methyl}-6-hydroxy-1,4-diazepan-1-yl)ethan-1-one
3-(3-fluoro-4-phenylbenzoyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidine
3-[(4-fluorophenyl)methyl]-5-[1-(2-methylbenzoyl)piperidin-4-yl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
N-(1H-imidazol-2-ylmethyl)-N-methyl-1-(2-phenylethyl)piperidin-3-amine
N-cyclopropyl-4-[1-(2-methoxyphenyl)piperidin-4-yl]piperazine-2-carboxamide
{1-methyl-4-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]piperazin-2-yl}methanol
3-(2-methoxybenzoyl)-1-[3-(5-methylfuran-2-yl)benzoyl]piperidine
1-{[4-(difluoromethoxy)phenyl]methyl}-4-(2-methylpyridin-4-yl)-1,4-diazepane
1-(2-phenylethyl)-4-[2-(trifluoromethyl)pyrimidin-4-yl]piperazin-2-one
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-2-ethoxybenzamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
N-ethyl-1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
(2R,3R)-3-amino-1'-(6-methyl-2-phenylpyrimidin-4-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
ethyl 1-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]-3-(3-phenylpropyl)piperidine-3-carboxylate
1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
(2E)-1-[4-(4-{[(1-benzothiophen-2-ylmethyl)(methyl)amino]methyl}phenoxy)piperidin-1-yl]-3-(4-methoxyphenyl)prop-2-en-1-one
8-(2-methyloxolane-2-carbonyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1-{[3-(cyclopentyloxy)phenyl]methyl}piperidin-4-yl)(1-methyl-1H-imidazol-2-yl)methanol
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}dimethylamine