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N-cyclopropyl-3-[5-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
4-(methoxymethyl)-1-{[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperidine
phenyl (3S,5R,9R)-5-hydroxy-2,8-dioxo-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-11-carboxylate
(3R,4R)-3-(azepan-1-ylmethyl)-N-cyclopentyl-4-(hydroxymethyl)pyrrolidine-1-carboxamide
N-(4-{1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1H-imidazol-2-yl}phenyl)acetamide
1-(7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-({7-[(5-ethylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
2-methyl-6-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane-8-carbonyl}-2,3-dihydropyridazin-3-one
8-(5-methoxyfuran-2-carbonyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
(1R,5R)-N,N-dimethyl-6-[2-(phenylsulfanyl)ethyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-(4-{[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]amino}piperidin-1-yl)-6-methylpyrimidin-2-amine
(1S,6R)-3-[(1-methyl-1H-indol-2-yl)methyl]-3,9-diazabicyclo[4.2.1]nonane
(1r,4r)-4-({[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)cyclohexan-1-ol
1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
N-(1H-1,3-benzodiazol-2-ylmethyl)-3-ethyl-5-hydroxyadamantane-1-carboxamide
N-[(7-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]thiophene-2-carboxamide
2-ethyl-4-{5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1-methylpiperazine
9-methoxy-10-(4-methylpiperazine-1-carbonyl)-3-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
5-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-[(3-methylpyridin-4-yl)methyl]-1,2-oxazole-3-carboxamide
methyl 5-({2-[2-(furan-2-yl)azepan-1-yl]acetamido}methyl)furan-2-carboxylate
2-(ethylamino)-N-[2-(3-methoxyphenyl)ethyl]pyrimidine-5-carboxamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
3-{[(butan-2-yl)(pyridin-3-ylmethyl)amino]methyl}-1-methyl-1,2-dihydroquinolin-2-one
2-[3-oxo-9-(5-oxopyrrolidine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-2-yl]acetic acid
methyl 5-[(3R)-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
1-ethyl-5-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
4-phenyl-1-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}azepane
2-({1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}methyl)-1H-1,3-benzodiazole
N,6-dimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
5-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-4-yl}-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
N-[(1S,2R)-2-carbamoylcyclopentyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-({3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]phenyl}methyl)propanamide
2-(dimethylamino)-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-4-methylpyrimidine-5-carboxamide
N-ethyl-2-[4-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenyl]acetamide
5-(1-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-1,2,3-triazol-4-yl)pyrimidine
1-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-methylbutan-1-one
N-(2-methoxyethyl)-N-[(2-methylphenyl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-[(3R,4S)-1-(1-acetylpiperidine-4-carbonyl)-4-cyclopropylpyrrolidin-3-yl]furan-3-carboxamide
4-{4-[(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)amino]piperidin-1-yl}-6-methylpyrimidin-2-amine
ethyl 1-[3-(1,2-oxazolidin-2-yl)propanoyl]-3-(3-phenylpropyl)piperidine-3-carboxylate
3-(piperidin-3-yl)-N-[2-(pyridin-4-yl)ethyl]benzamide
3-(2-oxo-2-{4-[(pyrimidin-2-yl)amino]piperidin-1-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(3-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(2R,3R)-2-ethoxy-1'-[(2-hydroxy-5-methoxyphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
1-[({5-propylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]cyclohexan-1-ol
6-fluoro-2-(pyrimidin-5-yl)-4-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]quinoline
2-fluoro-5-({[1-(methoxymethyl)cyclopentyl]carbamoyl}amino)-N-methylbenzamide
3-(1-ethyl-1H-imidazol-2-yl)-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]piperidine