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3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[(3-methylpyridin-4-yl)methyl]propanamide
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(3-methyloxetan-3-yl)methyl]acetamide
4-{5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}-1,4-oxazepane
(3S)-1-(1-methyl-5-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-1H-1,3-benzodiazol-2-yl)pyrrolidin-3-ol
1-(cyclohex-3-en-1-ylmethyl)-4-[2-(4-fluorophenoxy)ethyl]-1,4-diazepan-5-one
5-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]pyridine-2-carbonitrile
1-(morpholine-4-carbonyl)-4-(oxan-4-yl)-1,4-diazepane-6-carboxylic acid
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N-methyl-1H-1,3-benzodiazole-2-carboxamide
4-chloro-1,3-dimethyl-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]-1H-pyrazole-5-carboxamide
1-(2-hydroxypropanoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-{1-[1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)piperidin-4-yl]ethyl}morpholine
4-methyl-2-{2-[4-(2-methylpropyl)-3-oxo-6-(pyridin-2-ylmethoxy)-1,4-diazepan-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)(propan-2-yl)amine
1-(piperidin-1-yl)-2-(4-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazin-1-yl)ethan-1-one
3,3-dimethyl-1-({5-[(2,3,5-trifluorophenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
(1R,2R,6S,7S)-4-(6-phenylpyridazin-3-yl)-4-azatricyclo[5.2.1.02,6]decane
N-[2-(dimethylamino)ethyl]-4-[3-(trifluoromethyl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
2-(2,3-dihydro-1H-inden-1-yl)-1-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}ethan-1-one
4-(3-{7,9-dioxo-8-azaspiro[4.5]decan-8-yl}propoxy)benzamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-hydroxy-3-methylbutanamide
1-benzyl-4-[3-(methylsulfanyl)propyl]-1,4-diazepan-6-ol
2-(4-methoxyphenoxy)-1-{4-[2-(oxolan-2-yl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
3-(aminomethyl)-4-[(1S)-1-cyclohexylethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-ethyl-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]pyrimidin-2-amine
5-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidine-1-carbonyl]-3-methyl-2,3-dihydro-1,3-benzoxazol-2-one
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyrrolidine-1-sulfonamide
N-phenyl-5-(1,2,3,4-tetrahydroisoquinolin-5-yl)furan-2-carboxamide
4-[1-(2-fluorophenyl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]benzene-1-sulfonamide
1-(quinoline-5-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[2-(3,4-dimethoxyphenyl)propan-2-yl]-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
4-(4-methylbenzoyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2,3-difluoro-6-methoxy-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
3-[(1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)oxy]pyridine
(5-{[1-(4-methoxy-2,3-dimethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}furan-2-yl)methanol
8-(2,6-difluorobenzoyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(3S)-1-{4-methyl-6H,7H,8H-cyclopenta[g]quinolin-2-yl}pyrrolidin-3-yl]acetamide
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
1-[(2-chlorophenyl)methyl]-4-({thieno[2,3-d]pyrimidin-4-yl}amino)pyrrolidin-2-one
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-(1H-pyrazole-4-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
N-(2-methoxyethyl)-N,2,7-trimethylquinoline-4-carboxamide
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-{2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}ethan-1-one
2-(4-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl}piperidin-1-yl)acetamide
3-methyl-5-{4-[1-(morpholin-4-yl)ethyl]phenyl}pyridin-2-amine
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[2-(trifluoromethyl)phenyl]methyl}propanamide
4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1λ6-thiomorpholine-1,1-dione
9-[6-(trifluoromethyl)pyridin-2-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
6-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]imidazo[1,2-a]pyridine-2-carboxamide
3-({4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
8-fluoro-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]quinoline-2-carboxamide
1-[3-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenyl]ethan-1-one