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6-(2-fluoro-4-methoxyphenyl)-7-methyl-N-[2-(methylamino)ethyl]-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(3R,4S)-4-cyclopropyl-1-(3-phenoxypropyl)pyrrolidin-3-amine
2-{1-[2-(dimethylamino)ethyl]-3-(3-fluorophenyl)-2,5-dioxopyrrolidin-3-yl}-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]acetamide
N-[2,2-dimethyl-3-(morpholin-4-yl)propyl]pyrazin-2-amine
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-(pyridin-2-ylmethyl)benzamide
1-(cyclopropylmethyl)-3-(2-methylquinolin-5-yl)-6-(oxolane-2-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-{4-[4-(morpholin-4-yl)piperidin-1-yl]phenyl}-5-phenylpentanamide
6-[1-(4-cyclopentylpyrimidin-2-yl)piperidin-4-yl]-2-methylpyrimidin-4-ol
3-{4-[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]-1H-1,2,3-triazol-1-yl}propane-1,2-diol
2-{[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]methyl}-4-oxo-1,4-dihydroquinoline-6-carboxamide
9-(5-ethylthiophene-2-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2-{6-[(4-fluorophenyl)methoxy]-3-oxo-4-(propan-2-yl)-1,4-diazepane-1-carbonyl}phenyl)-1,3-diazinane-2,4-dione
1-(3-methylbutyl)-8-[3-(5-methylfuran-2-yl)butyl]-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 2-{2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}acetate
1-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-3-(1,2,3-thiadiazol-5-yl)urea
1-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-3,3-dimethylbutan-1-one
1-(4-{2-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]phenoxy}piperidin-1-yl)-2-methoxyethan-1-one
1-[4-(azepan-1-yl)-5-methylthieno[2,3-d]pyrimidine-6-carbonyl]-N,N-diethylpyrrolidin-3-amine
1-(cyclohexylmethyl)-4-oxo-N3-(propan-2-yl)-N5-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
5-[2-(benzylamino)ethyl]-1-(prop-2-en-1-yl)pyrrolidin-2-one
1-{2-[({4-[3-(4-ethylpiperazin-1-yl)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)amino]ethyl}pyrrolidin-2-one
N-(oxan-4-yl)-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carboxamide
N-cyclopropyl-3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
N-({3-methyl-7-[3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-carboxamide
N-[(3-tert-butyl-1,2,4-oxadiazol-5-yl)methyl]-6-(propan-2-yl)pyrimidin-4-amine
3-{5-[(2-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-(pyrrolidin-1-yl)propan-1-one
2-chloro-N-[2-({6-chloro-3-fluoroimidazo[1,2-a]pyridin-2-yl}formamido)ethyl]benzamide
N-{1-[1-(2,3-dimethoxybenzoyl)piperidin-4-yl]-2-phenylethyl}-2-(dimethylamino)-N-methylacetamide
2-(pyridin-4-yl)-N-{[4-(trifluoromethoxy)phenyl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]-1,2-oxazole-3-carboxamide
6,7-dimethoxy-2-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
(1S,5R)-3-[(2,3-dichlorophenyl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S)-2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-(2,6-dimethoxypyridin-3-yl)pyrrolidine-1-carboxamide
N-(4-{4-[(butan-2-yl)amino]piperidin-1-yl}phenyl)-2,4-dimethylbenzamide
N,1,3-trimethyl-N-[2-(morpholin-4-yl)propyl]-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
{1-[3-({[2-(cyclohex-1-en-1-yl)ethyl]amino}methyl)-7-methoxyquinolin-2-yl]piperidin-3-yl}methanol
N-methyl-5-{4-[4-(4-methylphenyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}pyrimidin-2-amine
3-(2H-1,3-benzodioxol-5-yl)-N-[2-(dimethylsulfamoyl)ethyl]-3-phenylpropanamide
N,1,3-trimethyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
1-{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-3-(1H-imidazol-1-ylmethyl)piperidine
N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-(1H-pyrazol-1-yl)butanamide
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-2-methylimidazo[1,2-a]pyridine-6-carboxamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
2-[({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]-N-methylpyridine-3-carboxamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-1-methyl-6-oxopiperidine-3-carboxamide
2-methoxy-N-[1-methyl-7-(4-propylpiperazine-1-carbonyl)-2-(pyridin-4-yl)-1H-1,3-benzodiazol-5-yl]acetamide
2-{4-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]piperidin-1-yl}acetamide
N-[(3-ethoxyphenyl)methyl]-N-(prop-2-en-1-yl)-2-(1H-1,2,4-triazol-1-yl)acetamide
2-[1-(azepane-1-sulfonyl)pyrrolidin-2-yl]-1-methyl-1H-1,3-benzodiazole
2-methyl-N-(oxan-4-yl)-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine