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3-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carbonyl}-6-(propan-2-yl)-1,2-dihydropyridin-2-one
N-cyclohexyl-N-[(4-methoxy-2,5-dimethylphenyl)methyl]-2-(4-methyl-2-oxopyrrolidin-1-yl)acetamide
2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}acetamide
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-2-(methoxymethyl)-N,1-dimethyl-5-(2-phenylacetamido)-1H-1,3-benzodiazole-7-carboxamide
9-(3-fluoro-4-methoxybenzenesulfonyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
1-methyl-4-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}piperazine
N-{1-[1-(1-phenoxypropan-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
3-methyl-N-({1-[(2E)-2-methylpent-2-en-1-yl]pyrrolidin-3-yl}methyl)furan-2-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
2-[3-(2-fluorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-[1-(4-methoxyphenyl)ethyl]-N-methylacetamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2,7-dioxo-1,3-diazepane-4-carboxamide
6-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2-methyl-1,3-benzoxazole
2,3-dimethyl-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]quinoxaline-6-carboxamide
N-butyl-N-(furan-2-ylmethyl)-6-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
(1R,3S)-7-{6-chloro-3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-7-azaspiro[3.5]nonane-1,3-diol
8-(2H-1,3-benzodioxol-5-ylmethyl)-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[1-(3-chlorobenzoyl)piperidin-3-yl]-N-[(2,4-dimethoxyphenyl)methyl]propanamide
(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amine
1-[(5-ethylpyridin-2-yl)methyl]-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]furan-2-carboxamide
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3H,4H-pyrido[2,3-d]pyrimidin-4-one
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-methoxyphenyl)methyl]acetamide
(5S,9aS,9bS)-5-(2,1,3-benzothiadiazol-5-yl)-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
7-[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazole-4-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-(2-ethoxyethyl)-5-(4-methyl-3-oxopiperazine-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-{[4-(difluoromethoxy)phenyl]methyl}-3-(2-methoxyphenoxy)azetidine
2-methoxy-N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
N,N-dimethyl-3-[({2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)methyl]benzamide
methyl 3-[(3S,4R)-1-[(2-ethoxyphenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]propanoate
N-{[7-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-2-sulfonamide
N-(1-methyl-1H-pyrazol-3-yl)-2-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-2-(2,4-dioxoimidazolidin-1-yl)acetamide
4-[(2-methyl-1H-imidazol-1-yl)methyl]-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidine
(2E)-3-(4-methoxyphenyl)-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)prop-2-enamide
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-6-methoxy-1-methyl-1H-indole-2-carboxamide
[4-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol
N-(furan-2-ylmethyl)-3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-(pyridin-4-ylmethyl)propanamide
ethyl 4-[2-(2-{[(2-fluorophenyl)methyl]amino}ethyl)-5-oxopyrrolidin-1-yl]piperidine-1-carboxylate
N-ethyl-6-fluoro-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(2-methylpyrimidin-5-yl)quinoline-4-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-ol
2-{2,8-diazaspiro[4.5]decan-2-yl}-1,3-thiazole-4-carboxamide
N-[(3R,4R)-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
8-[(3-hydroxyphenyl)methyl]-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)-2-(thiophen-3-yl)acetamide
N-{[2-(2,5-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-4-methylbenzamide
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-[(2-fluorophenyl)methyl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide