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N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclopentanecarboxamide
N,2-dimethyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-6-(4-methoxyphenyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
5-cyclopropanecarbonyl-1'-(2-ethylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-{[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzoic acid
methyl 9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-3-[(5-methylthiophen-2-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(1-propylpiperidin-4-yl)pyrrolidin-3-yl]acetamide
5-[2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)butanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
N-methyl-3-(methylsulfanyl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]propanamide
(2S,4R)-4-amino-1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-[2-(2-chloro-4-fluorophenyl)acetyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
N,N,4-trimethyl-5-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]pyrimidin-2-amine
1-[(3S,4S)-3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]pyrrolidin-1-yl]-4-methylpentan-1-one
ethyl 1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
(3S,4R)-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-ethyl-2-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine
3-[3-(cyclopropylmethyl)-1-[(4-ethylphenyl)methyl]-1H-1,2,4-triazol-5-yl]-N,N-dimethylpropanamide
2-(4-methyl-1H-pyrazol-1-yl)-1-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propan-1-one
8-fluoro-3-{2-[1-(propan-2-yl)piperidin-2-yl]ethyl}-3,4-dihydroquinazolin-4-one
1-[2-chloro-4-(1H-pyrazol-1-yl)benzoyl]-3-(hydroxymethyl)piperidin-3-ol
3-(2-chlorophenyl)-1-(3-hydroxyazetidin-1-yl)-3-phenylpropan-1-one
(4aS,7aR)-1-[2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
5-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
6-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
(2R,6R)-1-(1-cycloheptyl-1H-1,2,3-triazole-4-carbonyl)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
4-{4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]piperidine-1-carbonyl}pyridazine
1-benzyl-3-(pyridin-2-ylmethyl)-8-[(2,4,5-trimethylphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(cyclopropylmethyl)-5-(1H-indole-2-carbonyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-(1,2-oxazinan-2-yl)pyridine-3-carboxamide
3-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
(3aR,6aR)-N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-(2-chlorophenyl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-phenylpropanamide
4-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,3-thiazole-4-carbonyl)piperidine
ethyl 2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}-1,3-oxazole-4-carboxylate
5-{1-[(3-chlorophenyl)methyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-oxo-2,3-dihydro-1H-indene-1-carboxamide
3,4,5-trimethoxy-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzamide
(2S)-2-acetamido-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(methylsulfanyl)butanamide
(4aS,7aR)-1-(1H-imidazol-2-ylmethyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(pyridin-3-yl)-4-{[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]methyl}benzamide
3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-[3-(morpholin-4-yl)propyl]propanamide
2-[(3-fluorophenyl)methyl]-4-{4-[3-(trifluoromethyl)benzoyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
2-methylpropyl N-methyl-N-({1-[(3R,5S)-5-(methylcarbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazol-4-yl}methyl)carbamate
methyl 4-({[(3S,5S)-1-(2,3-dihydro-1H-inden-2-yl)-5-[(pyridin-3-ylmethyl)carbamoyl]pyrrolidin-3-yl]amino}methyl)benzoate
(1R,5S)-6-({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)-6-azabicyclo[3.2.1]octane
4-{[7-chloro-2-(thiophen-3-yl)quinolin-3-yl]methyl}piperazin-2-one