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1-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-(3-methylpyridin-4-yl)-1,4-diazepane
5-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-2-(furan-2-yl)pyrimidine
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-{4-[(2-methylbutyl)amino]piperidin-1-yl}benzamide
5-methanesulfonyl-1'-(oxan-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-{3-[3-(4-fluorophenyl)pyrrolidin-1-yl]-3-oxopropyl}-5-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidin-2-one
(4aS,7aR)-1-(2-methoxypyridine-4-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-{1-[2-(3-methylphenyl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
N-methyl-2-[3-(1H-pyrazol-5-yl)phenyl]pyridine-3-carboxamide
3-methyl-4-({2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-amino-4-[2-(piperidin-1-yl)pyrimidin-5-yl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
1-(cyclopropylmethyl)-5-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[(3R,4R)-1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
(2R,3R)-1'-(4-aminopyridine-2-carbonyl)-3-(dimethylamino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]-1H-indole-6-carboxamide
3-(5-chloro-2-methoxybenzoyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
3-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]-1H-pyrazol-5-amine
N-cyclopropyl-3-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}propanamide
2-(cyclohexylmethyl)-4-(1,2,3-thiadiazole-4-carbonyl)morpholine
N-(3-ethoxypropyl)-2-{2-[(4-phenylpiperazin-1-yl)methyl]-4-(thiophen-3-yl)phenoxy}acetamide
4-chloro-2-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}phenol
N-methyl-3-(2-phenylethyl)-N-[1-(1,3-thiazol-2-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
1-[(2S)-oxolan-2-ylmethyl]-2-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazole
2-[1-(cyclopropylmethyl)-4-(2-ethylpyrimidine-5-carbonyl)piperazin-2-yl]ethan-1-ol
1-propyl-4-[(5-{pyrazolo[1,5-a]pyridin-2-yl}-1,2,4-oxadiazol-3-yl)methyl]piperidine
N-(3,4-dimethoxyphenyl)-1-(1H-imidazol-4-ylmethyl)piperidin-3-amine
6-({3-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)quinoline
(2,1,3-benzoxadiazol-5-ylmethyl)[1-(1H-imidazol-1-yl)propan-2-yl]amine
N-methyl-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)propanamide
3-methyl-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)benzamide
[(2S,4R,5R)-5-(4-chlorophenyl)-4-({[(4-ethoxyphenyl)methyl]amino}methyl)-1-ethyl-2-methylpyrrolidin-2-yl]methanol
2-(dimethyl-1,3-thiazol-4-yl)-N-[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]acetamide
3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[1-(pyrazin-2-yl)propan-2-yl]benzamide
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-(propan-2-yloxy)pyrimidin-2-amine
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}[(5-fluoro-1H-indol-2-yl)methyl]methylamine
2-amino-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-4-(trifluoromethyl)pyrimidine-5-carboxamide
N'-(3,5-dimethylphenyl)-N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]propanediamide
9-(4-amino-3-hydroxybutanoyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
[(3R,4R)-1-(5-chloro-2-methylbenzoyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
(1S,5R)-3-(oxan-4-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1R,9S)-11-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
(1S,2S)-N2-(1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-2,3-dihydro-1H-indene-1,2-diamine
1-cycloheptyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-6-oxopiperidine-3-carboxamide
4-{1-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1H-imidazol-2-yl}benzoic acid
1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(pyridin-2-yl)ethan-1-one
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-3-(2-oxoazepan-1-yl)propanamide
N-({8-[(2-hydroxynaphthalen-1-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
3-[(4-ethylpiperidin-1-yl)methyl]-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
1-{1'-[(5-hydroxy-2-methoxyphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
2-[(2,4-dimethoxyphenyl)methyl]-4-{4-[2-(pyridin-3-yl)piperidine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione