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2-amino-4-ethyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-1,3-thiazole-5-carboxamide
1-[4-(2-chlorophenoxy)piperidin-1-yl]-2-(4-ethylpiperazin-1-yl)ethan-1-one
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-5-propyl-1,2-oxazole-3-carboxamide
1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propan-1-one
5-[1-(3-cyclopentylpropanoyl)piperidin-4-yl]-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
N-{[1-(4-ethenylbenzoyl)piperidin-3-yl]methyl}-1H-indole-2-carboxamide
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[3-(propan-2-yloxy)benzoyl]piperidine
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-3-(pyridin-3-yl)propanamide
1-{2-[ethyl(methyl)amino]acetyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(1R,7S)-6-(5-oxo-1,4-diazepane-1-carbonyl)-3-(2-phenoxyethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
11-[(cyclopropylmethyl)amino]-4-[(4-methylphenyl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-[1-(6-ethyl-2-methylquinoline-4-carbonyl)-3-oxopiperazin-2-yl]-N-methylacetamide
6-ethyl-3-(1H-imidazol-2-ylmethyl)-3,4-dihydroquinazolin-4-one
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidine
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
1-{2-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]phenyl}ethan-1-one
(3S,4R)-1-[4-(furan-2-yl)benzoyl]-4-methylpiperidine-3,4-diol
(2S)-2-amino-3-methoxy-N-[3-(2-phenylacetamido)phenyl]propanamide
2,3-dimethyl-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]quinoxaline-6-carboxamide
4-[3-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)benzenesulfonyl]piperazin-2-one
2-[({1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)(methyl)amino]-N-methylacetamide
(3S,5R)-N3-(2H-1,3-benzodioxol-5-ylmethyl)-N5-(2,3-dihydro-1H-inden-5-yl)-1-(naphthalen-2-ylmethyl)piperidine-3,5-dicarboxamide
4-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
(2S,4R)-4-amino-1-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methylpyrrolidine-2-carboxamide
N-[(3-methylthiophen-2-yl)methyl]-N-(oxolan-3-ylmethyl)cyclopropanamine
1-cycloheptyl-4-[(pyridin-4-ylmethyl)amino]pyrrolidin-2-one
(3S,4R)-1-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(5-methylhex-5-en-2-yl)amine
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[(1-methyl-3-phenyl-1H-pyrazol-5-yl)methyl]acetamide
3-cyclopropyl-6,7-dimethoxy-3,4-dihydroquinazolin-4-one
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
ethyl 4-[1-(5-methoxyfuran-2-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
1-ethyl-3-methyl-N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-1H-pyrazole-5-carboxamide
2-{[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-3,4-dimethoxypyridine
3-[4-(3,4-difluorophenyl)-1H-pyrazol-5-yl]-1-[(5-methylthiophen-2-yl)methyl]piperidine
2,4-difluoro-N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)benzamide
5-methyl-1-(3-methylphenyl)-4-(3-phenylbenzoyl)piperazin-2-one
N,N-dimethyl-3-[(quinolin-4-ylmethyl)sulfamoyl]benzamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)acetamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
6-fluoro-2-[(4-methyl-1,4-diazepan-1-yl)methyl]quinolin-4-ol
N,3,4-trimethyl-N-(prop-2-yn-1-yl)-5-sulfamoylbenzamide
N-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)acetamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
4-benzyl-1-[2-(2,3,4-trifluorophenyl)acetyl]-1,4-diazepan-5-one
2-amino-4-methyl-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrimidine-5-carboxamide
11-{[(3-fluorophenyl)methyl]amino}-4-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[4-benzyl-2-(hydroxymethyl)piperazin-1-yl]-4-(piperidin-1-yl)butan-1-one
9-{[2-(butan-2-yloxy)-3-methoxyphenyl]methyl}-2-methyl-2,9-diazaspiro[5.5]undecan-3-one