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(4S,6R)-4-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane-11-carbonyl}-6-methyl-1,3-diazinane-2-thione
3-(2-methoxyphenyl)-5-[(4-methylpiperazin-1-yl)sulfonyl]benzoic acid
1-({4-[(2,5-dimethylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-3-carboxamide
N-(pyridin-2-ylmethyl)-4-(thiophen-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[2-(4-methoxyphenyl)phenyl]-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidine-3-carboxamide
N-[2-(3-phenylpiperidin-1-yl)ethyl]-1H-imidazole-2-carboxamide
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-4-oxo-4H-chromene-2-carboxamide
1-{[2-(benzylamino)pyrimidin-5-yl]methyl}azetidin-3-ol
3-{2-hydroxy-N-methyl-2-[4-(trifluoromethyl)phenyl]acetamido}-N-methylpropanamide
(4S,4aS,8aS)-1-[(3-methylpyrazin-2-yl)methyl]-4-phenyl-decahydroquinolin-4-ol
1-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-(1H-imidazol-1-yl)ethan-1-one
2-({2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}methyl)benzonitrile
N-{1-[7-(2,6-dimethoxybenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}-2-(dimethylamino)acetamide
4-methylphenyl (7S,9aR)-7-(cyclohexylmethyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
methyl 4-{[3-(2-methoxybenzoyl)piperidine-1-carbonyl]amino}benzoate
2-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
2-(4-cyclohexyl-1,4-diazepan-1-yl)pyridine-4-carboxylic acid
2-[3-(4-methoxyphenyl)-4-methyl-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
5-(4-cyclohexylphenyl)-N-(1,4-dioxan-2-ylmethyl)-1,2,4-triazin-3-amine
[(2R)-1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl]methanol
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}[(6-methylpyridin-2-yl)methyl](oxolan-2-ylmethyl)amine
3-{2-[3-(2-ethoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
N4-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-5-ethylpyrimidine-2,4-diamine
N,N,4-trimethyl-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrimidin-2-amine
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[4-(1H-pyrazol-1-yl)butan-2-yl]propanamide
2-methyl-4-(3-{2-methyl-2,8-diazaspiro[4.5]decane-8-carbonyl}phenyl)butan-2-ol
1-(cyclopropylmethyl)-5-(2-methyl-1,3-thiazole-4-carbonyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(2-methoxyphenyl)-4-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}piperazine
N-[3-(1H-indazol-1-yl)propyl]-4-sulfamoylbenzamide
6-chloro-N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(pyrimidin-5-yl)quinoline-4-carboxamide
5-(methoxymethyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
N-(3-acetamido-4-methoxyphenyl)-4-ethoxypiperidine-1-carboxamide
1-[4-(furan-2-ylmethyl)piperazin-1-yl]-3-(3-hydroxyquinoxalin-2-yl)propan-1-one
5-ethyl-N-[(4-fluorophenyl)methyl]-N-(1-hydroxybutan-2-yl)thiophene-2-carboxamide
N-[(4-fluorophenyl)methyl]-4-hydroxy-N-methyl-2-(4-methylphenyl)pyrimidine-5-carboxamide
3-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-N,N-dimethylaniline
3-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)phenol
1-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-3-(1-methyl-1H-1,2,3-benzotriazol-5-yl)urea
methyl 3-(oxolane-3-amido)-1-(2-phenylethyl)-5-{[1-(pyridin-3-yl)propan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
8-[2-(4-fluorophenoxy)ethyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 2-[(2,3-dimethylphenyl)sulfamoyl]-6-(2-methylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3,5-dichloro-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-4-(prop-2-en-1-yloxy)benzamide
N-cyclopropyl-2-(morpholin-4-yl)-6-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}pyridine-3-carboxamide
5-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-3-(furan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(3S)-1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperidin-3-amine
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}[(4-fluorophenyl)methyl]methylamine
5-chloro-N-{2-[1-(2-methylpropyl)piperidin-3-yl]ethyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
2-benzyl-8-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[1-(1H-pyrrole-3-carbonyl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1H-pyrrole-3-carboxamide