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[(1-ethyl-1H-imidazol-2-yl)methyl]bis(1,3-oxazol-4-ylmethyl)amine
methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl][3-(piperidin-1-yl)propyl]amine
[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-3-(2-phenoxyethyl)piperidin-3-yl]methanol
N-{[1-(thian-4-yl)piperidin-3-yl]methyl}-3-(trifluoromethyl)benzamide
N-[2-methyl-5-({[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]carbamoyl}amino)phenyl]propanamide
1-{5-[6-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carbonyl]thiophen-2-yl}ethan-1-one
5-(3-methoxyphenyl)-3-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-1,2,4-triazine
1-cycloheptyl-6-oxo-N-[4-(pyridin-2-yl)butyl]piperidine-3-carboxamide
ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
7-fluoro-3-[(2-methylpiperidin-1-yl)methyl]-1-(pyridin-4-ylmethyl)-1,2-dihydroquinolin-2-one
6-methyl-5-(3-oxopiperazine-1-carbonyl)-4-[2-(prop-2-en-1-yloxy)phenyl]-1,2,3,4-tetrahydropyrimidin-2-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}acetamide
4,5-dimethyl 1-[(3S,5S)-1-[(4-methoxy-3-methylphenyl)methyl]-5-[(quinolin-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(4aS,7aR)-1-(3-ethyl-1H-pyrazole-4-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl 1-[(4-methoxyphenyl)methyl]-5-(1-methyl-1H-pyrazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-{1-[2-(2-ethoxyphenoxy)ethyl]pyrrolidin-2-yl}pyridine
1-(adamantan-1-yl)-4-(2-methyl-1,3-thiazole-4-carbonyl)piperazine
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2-(thiophen-2-yl)acetamide
1-[2-(4-fluoropiperidin-1-yl)-2-oxoethyl]-4-phenylpyrrolidin-2-one
N-({7-[(4-ethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzenesulfonamide
2-{1-ethyl-2,4-dioxo-8-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
5-{2-oxo-2-[4-(2-phenylethyl)piperidin-1-yl]ethyl}imidazolidine-2,4-dione
1-ethyl-N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
2-amino-4-[4-hydroxy-3-(prop-2-en-1-yl)phenyl]-6-(pyridin-3-yl)pyridine-3-carbonitrile
2-(4-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidine
3-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]naphthalen-2-ol
2-{5-[5-(oxolan-2-yl)thiophene-2-carbonyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
2-[5-cyclopropyl-4-(4-methylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-(furan-2-yl)pyrimidine
1-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-imidazol-1-yl)ethan-1-one
N-[1-(furan-2-yl)ethyl]-9-methoxy-3-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-{1-[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
N-(2-methoxyethyl)-1,3-dimethyl-N-(pyridin-4-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[(3-methylpyridin-4-yl)methyl]benzamide
(1S,5R)-6-[(4-methoxy-3-methylphenyl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-{5-[1-(4-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-2-methylphenyl}imidazolidin-2-one
N-[1-(thian-4-yl)piperidin-4-yl]-2,3-dihydro-1H-indene-1-carboxamide
5-{2-[4-(5-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
(3R,4S)-1-[1-(2-fluorophenyl)cyclopropanecarbonyl]-4-propylpyrrolidin-3-amine
5-(7-methoxy-2H-1,3-benzodioxol-5-yl)-4-phenyl-1H-imidazole
1-(3-cyanophenyl)-3-{[1-(propan-2-yl)piperidin-3-yl]methyl}urea
5-[(isoquinolin-5-yloxy)methyl]-N-(1-methoxybutan-2-yl)-1,2-oxazole-3-carboxamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]acetamide
2,4-dimethyl-3-oxo-N-[4-(thiophen-2-ylmethoxy)phenyl]piperazine-1-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2,3,4-trimethoxybenzamide
N-{[3-(furan-2-ylmethoxy)-4-methoxyphenyl]methyl}-N-(oxolan-2-ylmethyl)-3-(1H-pyrazol-1-ylmethyl)benzamide
1-(2-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}pyrimidin-4-yl)pyrrolidin-3-ol
1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-3-[4-(methylsulfanyl)benzoyl]piperidine
3-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzonitrile