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{3-[(2-fluorophenyl)methyl]-1-[1-(2-fluorophenyl)piperidin-4-yl]piperidin-3-yl}methanol
3-[2-(azocan-1-yl)-2-oxoethyl]-4-benzylpiperazin-2-one
3-(1H-imidazol-2-yl)-N-[1-(2-methoxyphenoxy)propan-2-yl]benzamide
N-[(3,4-difluorophenyl)methyl]-3-{1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-3-yl}propanamide
8-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-2,8-diazaspiro[4.5]decan-3-one
1-[3-({[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amino)propyl]pyrrolidin-2-one
2-{8-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
2-methoxy-N-methyl-5-({[(3R)-piperidin-3-yl]carbamoyl}amino)benzamide
1-(2-ethoxyethyl)-N-methyl-N-(1-methylpiperidin-4-yl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
5-[1-(3-fluorobenzoyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
(4aS,8aR)-6-(1-aminocyclobutanecarbonyl)-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
N-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}pyrazin-2-amine
methyl 3-acetamido-1-ethyl-5-({[2-(furan-2-yl)phenyl]methyl}amino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-[(2-{2-[4-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)sulfanyl]-1H-1,2,4-triazole
3-(4-hydroxyphenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
3-cyclopropyl-1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
4-{4-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(thiophen-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-3-(pyridin-3-yl)propan-1-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-{[4-(trifluoromethyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)propanamide
N-[2-chloro-5-(diethylcarbamoyl)phenyl]-6-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
1-{3-[3-(2-hydroxyethyl)-4-methylpiperazine-1-carbonyl]phenyl}imidazolidin-2-one
3-chloro-N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-4-fluoro-1-benzothiophene-2-carboxamide
N-methyl-2-{[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}pentanamide
1-[(4aS,8aS)-4a-hydroxy-7-[4-(pyrrolidin-1-yl)benzoyl]-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
methyl 9-[2-(2-fluorophenyl)ethoxy]-3-[(3-hydroxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-fluoro-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
6-[(1-methyl-1H-indol-3-yl)methyl]-4-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
2-phenyl-N-({7-[(4-phenylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
(3S,4R)-4-(3-methylthiophen-2-yl)-1-(quinoline-4-carbonyl)piperidin-3-ol
5-{2-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(4-chlorophenyl)-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-3-phenylpropanamide
4-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-1-(4-methylphenyl)piperazin-2-one
(1R,6S)-9-methyl-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-3,9-diazabicyclo[4.2.1]nonane
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
N-methyl-N-[(6-methylpyridin-2-yl)methyl]-1-(2-phenylethyl)piperidin-3-amine
2-(1H-pyrrol-1-yl)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)propanamide
N,N-diethyl-1-[(1s,4s)-4-cyclobutaneamidocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-2-methyl-4,5,6,7-tetrahydro-1-benzofuran-4-one
N-(furan-2-ylmethyl)-2-{3-[3-(6-methylpyridin-3-yl)phenyl]-1H-pyrazol-1-yl}acetamide
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-4-(pyridin-2-yl)pyrimidin-2-amine
1-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)piperidin-4-ol
2-(7-methyl-1H-indol-3-yl)-1,3-thiazole-4-carboxamide
7-(5-chloropyridin-2-yl)-4-(cyclopropylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(2-chlorophenyl)methyl]-N-methyl-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
(2S)-2-[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]-4-methylpentanamide
N-[6-(2-aminoethyl)pyrimidin-4-yl]-1-phenyl-3,6-diazatricyclo[4.3.1.13,8]undecan-9-amine