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3-[2-(3-acetylpiperidin-1-yl)-2-oxoethyl]-1-cyclopropyl-3-(4-methoxyphenyl)pyrrolidine-2,5-dione
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
6-ethoxy-4-methyl-2-[4-(quinolin-2-ylmethyl)-1,4-diazepan-1-yl]quinazoline
1-methyl-4-(1,2,3,4-tetrahydroquinoline-8-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(2-methoxyethyl)-1-methyl-2-oxo-N-(pyridin-3-ylmethyl)-1,2-dihydroquinoline-4-carboxamide
1-(3-fluorophenyl)-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-pyrazole
(1R,5R)-N,N-dimethyl-6-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propanamide
4-(1H-pyrazol-4-yl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}butan-1-one
N-(2-hydroxyethyl)-4-{methyl[2-(oxan-2-yl)ethyl]amino}pyridine-2-carboxamide
N-methyl-2-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidin-4-amine
2-(ethylamino)-5-methyl-N-{[6-oxo-2-(pyrazin-2-yl)-1,6-dihydropyrimidin-4-yl]methyl}benzamide
1-methyl-3-{4-[(4-methylphenyl)methyl]-3-oxopiperazine-1-carbonyl}-1,2-dihydroquinolin-2-one
3-(2,1,3-benzothiadiazol-5-ylmethyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
3-ethyl-8-(4-oxo-1,4-dihydroquinoline-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(cyclopropylsulfamoyl)-5-(quinolin-5-yl)benzoic acid
9-[(2-aminopyridin-3-yl)methyl]-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
(3R,5S)-N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
ethyl 4-(cyclopropylmethyl)-1-(quinolin-6-ylmethyl)piperidine-4-carboxylate
{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
2-({[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}amino)pyridine-3-carbonitrile
4-methyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-3-(2-oxoimidazolidin-1-yl)benzamide
N-methyl-N-{1-[1-(4-methylpentanoyl)piperidin-4-yl]-2-(2-methylphenyl)ethyl}-2-(1H-pyrazol-1-yl)acetamide
N,2,5-trimethyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(1,3-thiazol-4-yl)ethyl]propanamide
N-(1-{7-[(3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylfuran-3-carboxamide
N-[(2R,3R)-1'-(5-propyl-1,2-oxazole-3-carbonyl)-2-(pyridin-4-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
1-(4-methylphenyl)-4-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)pyrrolidin-2-one
7-[(3-methylphenyl)methyl]-2-(prop-2-ene-1-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
4-(2,2-dimethyl-2,3-dihydro-1-benzofuran-7-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
methyl (2S)-1-(3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanoyl)pyrrolidine-2-carboxylate
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-[(1-methylpyrrolidin-3-yl)methyl]propanamide
3-(3-chlorophenyl)-5-[2-(1H-pyrazol-4-yl)ethyl]-1,2,4-oxadiazole
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(3-methylbutyl)-2,7-diazaspiro[4.5]decan-6-one
1-(furan-3-carbonyl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
1-(4-methoxybenzoyl)-4-[3-(5-methylfuran-2-yl)butyl]piperazine
(2S,4S)-4-amino-1-[6-(3-fluorophenyl)pyridine-3-carbonyl]pyrrolidine-2-carboxylic acid
4-benzyl-3-ethyl-1-(2-methylpyridine-3-carbonyl)-1,4-diazepan-5-one
1-(dimethyl-1,3-thiazole-5-carbonyl)-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N,N-diethyl-2-{[2-oxo-1-(2-phenylethyl)-4-(1,3-thiazole-4-carbonyl)-1,4-diazepan-6-yl]oxy}acetamide
4-(5-methylpyridin-2-yl)-1-{[2-(propylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-ol
N-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
2-[3,5-dimethyl-4-(3,3,3-trifluoro-2-methoxy-2-phenylpropanamido)-1H-pyrazol-1-yl]acetic acid
5-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}pyrimidine
3-(2,5-dimethoxyphenyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}pyrrolidine
3-[1-(3-chloro-4-fluorobenzoyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
N-[1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-yl]pyridin-2-amine
2-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
(1S,5R)-3-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
6,8-dimethoxy-4-methyl-N-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]quinolin-2-amine