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N-[(2,3-difluorophenyl)methyl]-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-methyl-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]propanamide
2-(4-methanesulfonylphenyl)-1-[2-methoxy-2-(thiophen-2-yl)ethyl]-1H-imidazole
1-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}azepan-4-amine
1-(3-methyl-5-propyl-1-benzofuran-2-carbonyl)piperidin-4-ol
5-methyl-N-[2-(2-methylpropanesulfonyl)ethyl]-1-propyl-1H-pyrazole-4-carboxamide
1-(1,2-benzoxazol-6-yl)-3-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}urea
N-{[8-(furan-3-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-2-phenylacetamide
2-methoxy-2-phenyl-N-{1-[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
N-{1-[7-(9H-fluoren-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-3-methoxypropanamide
2-(1-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-3-oxopiperazin-2-yl)-N-methylacetamide
5-[2-(2-methyl-1H-indol-3-yl)acetyl]-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl 5-[(4-oxo-4H-chromen-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
6-[1-(2,6-dimethylphenoxy)propan-2-yl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-(adamantan-1-yl)-1-[3-(pyridin-3-yl)azetidin-1-yl]ethan-1-one
methyl N-{[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})carbamoyl]methyl}carbamate
6-oxo-1-(2-phenylethyl)-N-[2-(1,3-thiazol-2-yl)ethyl]piperidine-3-carboxamide
(2S,4R)-1-(2-{[(2-chlorophenyl)methyl]sulfanyl}acetyl)-4-hydroxypyrrolidine-2-carboxylic acid
5-[1-(2,3-dimethylbenzoyl)piperidin-4-yl]-5-[(4-fluorophenyl)methyl]-3-(oxolan-3-yl)imidazolidine-2,4-dione
5-(1H-imidazol-1-ylmethyl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]furan-2-carboxamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
N-cyclopentyl-1-[(4-methoxyphenyl)methyl]-5-(1,2,5-thiadiazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]piperidin-3-ol
3-cyclopropyl-1-[4-(3-methylpyridin-4-yl)phenyl]urea
methyl 3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-2-ylmethyl)piperidin-3-yl]propanoate
2-cyclopropyl-1-[1-(pyridin-2-ylmethyl)-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
N-[(4-hydroxyazepan-4-yl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
3-{1-[(3,7-dimethyl-1H-indol-2-yl)methyl]piperidin-3-yl}-N-[(5-methylfuran-2-yl)methyl]propanamide
3-(2,6-dimethylphenoxy)-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}azetidine
{3-[(3-chlorophenyl)methyl]piperidin-3-yl}methanol
2-(3-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)quinoline
(3S)-3-({[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)azepan-2-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(2-hydroxyphenyl)acetamide
4-(2,3-dihydro-1H-isoindole-2-carbonyl)-2,6-dimethylquinoline
ethyl 5-{[4-(4-methyl-1,4-diazepan-1-yl)-6-oxo-1,6-dihydropyridazin-1-yl]methyl}furan-2-carboxylate
7-(3-chlorophenyl)-4-(2,5-dimethylfuran-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-cyano-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}benzamide
N-{3-[ethyl(phenyl)carbamoyl]phenyl}-2,6-dimethylpyrimidine-4-carboxamide
(2S)-2,6-diamino-N-(2-methoxy-5-{[1,3]oxazolo[4,5-b]pyridin-2-yl}phenyl)hexanamide
(4aS,7aR)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,5R)-6-(2-propyl-1,3-thiazole-4-carbonyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-{5-[3-(5-methylfuran-2-yl)butyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
8-cyclopropanecarbonyl-2-(2-methylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[2-(7-{[4-(dimethylamino)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-2-methylpropanamide
4-acetyl-5-butyl-1-(3-phenylphenyl)piperazin-2-one
6-[4-(quinolin-2-ylmethyl)piperazin-1-yl]pyridine-3-carboxamide
8-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-[2-(dimethylamino)ethyl]-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-(2-oxopyrrolidin-1-yl)-N-(pyridin-3-ylmethyl)acetamide
N-({7-[2-(2,5-dimethoxyphenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
2-(3-methyl-1H-pyrazol-1-yl)-N-[(2-phenoxypyridin-3-yl)methyl]acetamide