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1-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(1-methyl-1H-imidazol-2-yl)piperidine
(1S,5R)-6-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}-3-methyl-3,6-diazabicyclo[3.2.2]nonane
5-{[4-(2-methoxybenzoyl)piperazin-1-yl]methyl}-N,N-dimethylpyrimidin-2-amine
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
1-[2-(3,5-dimethoxyphenyl)ethyl]-2-(1H-imidazol-2-yl)-1H-imidazole
3-{2-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-oxoethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(4-fluoro-2-methylphenyl)-2-[(3-phenyl-1H-pyrazol-4-yl)formamido]propanamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-(2-methoxyethyl)-N-(propan-2-yl)benzamide
N-(3-ethoxypropyl)-1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(thiophen-2-yl)-1H-pyrazole-4-carboxamide
3-(2-hydroxyphenyl)-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-1H-pyrazole-5-carboxamide
(2S,4S)-N-ethyl-4-(2-methoxyacetamido)-1-[2-(3-methylphenyl)acetyl]pyrrolidine-2-carboxamide
4-[2-(1H-pyrazol-1-yl)ethyl]-1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine
N-(1-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
2-{3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]piperidin-1-yl}pyridine
2-{2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl}-2-azaspiro[4.5]decan-3-one
(3aS,6aS)-2-(2-hydroxyethyl)-5-(1H-indol-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
1-(3-chlorophenyl)-4-[1-(thiophene-3-carbonyl)piperidin-3-yl]piperazine
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
5-[3-(1,3-benzoxazol-2-yl)piperidine-1-carbonyl]-2-cyclopropylpyrimidin-4-ol
(1R,5S,6S)-N-cyclopentyl-3-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
5-{[3-(3-chlorophenyl)pyrrolidin-1-yl]methyl}-3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazole
4-{4-methoxy-3-[(methylamino)methyl]phenyl}-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-{4-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]piperazin-1-yl}pyrazine
4-[(2-benzoyl-1-benzofuran-3-yl)methyl]-1,4-oxazepan-6-ol
4-(3-fluoro-4-methoxyphenyl)-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}-1-(pyridin-4-ylmethyl)piperidin-4-amine
2-(morpholin-4-yl)-1-[3-(morpholine-4-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(2-methoxyethyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-benzoxazole-6-carboxamide
(1S,5R)-6-(2-fluoro-4-methylbenzoyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-2,4-dimethyl-1,3-thiazole-5-carboxamide
N-[(2,3-dimethoxyphenyl)methyl]-6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
5-(2-oxo-2-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}ethyl)-3-propylimidazolidine-2,4-dione
N-[(3S,4R)-4-(4-methylphenyl)-1-(quinoline-3-carbonyl)pyrrolidin-3-yl]acetamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)pyrazolo[1,5-a]pyridine-7-carboxamide
1-(furan-2-ylmethyl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
5-({5-[5-(oxolan-2-yl)thiophen-2-yl]-4-phenyl-1H-imidazol-1-yl}methyl)-1H-1,2,4-triazole
(1R,9aR)-1-({methyl[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
2-{4-[(2-fluorophenyl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
(1R,2R)-N-[2-(dimethylamino)ethyl]-2-phenyl-N-(thiophen-3-ylmethyl)cyclopropane-1-carboxamide
(2-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)urea
3-(1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carbonyl)pyridine
2-hydroxy-N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)propanamide
6-methyl-4-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-(cyclopent-2-en-1-yl)-N-cyclopropyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
6-{3-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
2-methyl-4-{3-[4-(pyridin-2-ylmethyl)piperazine-1-carbonyl]phenyl}butan-2-ol
N-ethyl-3-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propanamide