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2,2-dimethylpropyl N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}carbamate
N,4-dimethyl-N-{2-[2-(prop-2-en-1-yl)phenoxy]ethyl}pyridine-3-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,4-dimethyl-1,3-oxazole-5-carboxamide
(2S)-2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-4-methylpentanamide
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}({2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl})amine
4-(4-methylpiperazin-1-yl)-6-{4-[1-(morpholin-4-yl)ethyl]phenyl}pyrimidin-2-amine
1-(5-amino-4-chloro-1H-pyrazole-3-carbonyl)-3-ethylpiperidine-3-carboxamide
4-(1H-imidazol-2-yl)-1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)piperidine
3-ethyl-1-[3-(5-methylfuran-2-yl)benzoyl]piperidine-3-carboxylic acid
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-ethyl-4-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]methyl}-3,5-dimethyl-1H-pyrazole
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
3-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]pyridin-1-ium-1-olate
N-butyl-3-{[3-(pyridin-3-yl)azetidin-1-yl]sulfonyl}benzamide
[1-(7-fluoro-3-{[(2-phenylethyl)amino]methyl}quinolin-2-yl)piperidin-3-yl]methanol
N-[(2R,4R,6S)-2-cyclohexyl-6-(1-methyl-1H-imidazol-2-yl)oxan-4-yl]benzamide
3-{[3-(aminomethyl)pyrrolidin-1-yl]sulfonyl}-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]benzamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
2-cyclopentyl-1-{4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
4-(1-acetylpiperidin-4-yl)-1-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine
2-{[4-(5-chloropyrimidin-2-yl)piperazin-1-yl]methyl}-3-methoxyphenol
(2S)-2-amino-N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(1H-imidazol-4-yl)propanamide
1-{1-[(3-fluoro-4-methylphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
5-phenyl-N-{2-[3-(trifluoromethyl)phenyl]ethyl}-1,2,4-triazin-3-amine
9-methoxy-4-[(4-methoxyphenyl)methyl]-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)[(2-methylpyridin-4-yl)methyl]amine
2-methyl-6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}-2,3-dihydropyridazin-3-one
N-(3,4-dimethoxyphenyl)-1-[2-(trifluoromethyl)benzoyl]piperidin-3-amine
N-(2,3-dihydro-1H-inden-2-yl)-5,6-dimethyl-N-propylpyridine-3-carboxamide
N-[(2-fluorophenyl)methyl]-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
1-[(3aS,6aS)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-octahydropyrrolo[2,3-c]pyrrol-5-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
ethyl 1-{3-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]-6-(thiophen-2-yl)pyridin-2-yl}piperidine-3-carboxylate
N-methyl-1-(9H-purin-6-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)piperidin-4-amine
methyl 3-{[1-(cyclopropylmethyl)-5-[3-(trifluoromethyl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
4-chloro-N-(3-hydroxy-3-phenylpropyl)-N-methyl-1H-pyrrole-2-carboxamide
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(2-methoxyphenyl)-2-methylpiperazine
N-{1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-2-phenylethyl}-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
1-[2-hydroxy-3-(4-{[(3-hydroxy-2,2-dimethylpropyl)amino]methyl}-2-methoxyphenoxy)propyl]piperidin-4-ol
N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
(2R,4S)-4-hydroxy-1-[3-(prop-2-en-1-yloxy)benzoyl]piperidine-2-carboxylic acid
1-(1-benzylpyrrolidin-3-yl)-2-(propan-2-yl)-1H-imidazole
3-[5-(benzylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(2,3-dimethoxyphenyl)methyl]piperidine
9-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-2-[3-(dimethylamino)propyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{2-[(2E)-3-(1H-imidazol-4-yl)prop-2-enoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide
N,3-dimethyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
5-(2-fluorophenoxymethyl)-N-[1-(pyridin-4-yl)propyl]-1H-pyrazole-3-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-(1H-indole-2-carbonyl)-N-methylpiperidin-3-amine
(4aS,7aR)-4-benzyl-N-(4-methylphenyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
ethyl 3-{[methyl(1,2-oxazol-3-ylmethyl)carbamoyl]methyl}morpholine-4-carboxylate