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1-[(1S,5R)-6-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-{3-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]phenyl}acetamide
2-{4-[1-(4-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]piperazin-1-yl}pyrazine
4-(5-methyl-1-benzofuran-2-carbonyl)-1-(4-methylphenyl)piperazin-2-one
2-[3-(4-methoxy-3,5-dimethylphenyl)phenoxy]acetamide
1-ethyl-3-(propan-2-yl)-N-{[1-(pyrrolidin-1-yl)cyclopentyl]methyl}-1H-pyrazole-5-carboxamide
3-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}-1-[3-(oxolan-3-yl)propyl]urea
N-{[7-(5-acetylthiophen-2-yl)-1H,2H-naphtho[2,1-b]furan-2-yl]methyl}-2,2-dimethyloxane-4-carboxamide
5-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoxaline
5-(2-hydroxy-3-methoxybenzoyl)-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-4-(4-fluorophenyl)-1,4-diazepane
2-ethyl-9-(2-methoxy-3-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2,3-dihydro-1H-inden-5-yl)-3-(2-ethoxyethyl)-5-(1H-imidazol-1-ylmethyl)-1H-1,2,4-triazole
4-(3-methylbut-2-en-1-yl)-3-{2-[4-(morpholin-4-ylmethyl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
1-(1,4-dioxan-2-ylmethyl)-5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazole
2-{2-[1-(furan-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrrol-1-yl}-1,3-thiazole
N2,N2,5,6-tetramethyl-N4-[2-(pyrazin-2-yl)ethyl]pyrimidine-2,4-diamine
5-[(dimethylamino)methyl]-N-(2-ethoxybutyl)furan-2-carboxamide
5-methanesulfonyl-1'-(pyridine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-({3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)-2,1,3-benzothiadiazole
methyl 3-(2-chloro-6-fluorobenzamido)-6-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(3-methyl-1H-indole-2-carbonyl)pyrrolidin-3-yl]methanol
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
1-methyl-5-{3-methyl-1-[5-(1-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]butyl}-1H-1,2,4-triazole
5-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)-5-(2-phenylethyl)imidazolidine-2,4-dione
N-ethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
2-[methyl({[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]-1-phenylethan-1-ol
13-(2-phenylethyl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-hydroxy-3-methylbutan-1-one
1-({3-[(2-chloro-6-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrrolidin-2-one
(3S,9aR)-3-(cyclohexylmethyl)-8-(4-fluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{[1-(2H-1,3-benzodioxol-5-yl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-N-[2-methyl-2-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
2-(1-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
(4aR,7aS)-1-cyclopropanecarbonyl-4-(1,2,4-oxadiazol-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(2-methoxyphenyl)methyl]-4-[4-(2-methylphenyl)-1H-imidazol-2-yl]pyrrolidin-2-one
(4aS,7aR)-1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3R)-1-(5-chloro-2-fluorobenzoyl)-3,4,4-trimethylpyrrolidin-3-ol
1-{1'-[(2-fluoro-4-methoxyphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-[(4-acetamidophenyl)methyl]-2-[(1-methanesulfonylpiperidin-4-yl)amino]acetamide
N-{2-[(4-methylphenyl)sulfanyl]ethyl}-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-3,4,5-trimethoxybenzamide
9-[3-(2-ethoxyethoxy)benzoyl]-3-oxa-9-azaspiro[5.5]undecane
2-{3-[(4-methanesulfonamidopiperidin-1-yl)methyl]phenoxy}acetamide
1-(2-cycloheptyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]piperidine-4-carboxamide
1-[(3,5-dichloropyridin-4-yl)methyl]-4-(1-methylpiperidin-4-yl)piperazine
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
6-ethoxy-4-methyl-2-(4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1,4-diazepan-1-yl)quinazoline