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5-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-N-(2-hydroxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
ethyl 3-[(3-chlorophenyl)methyl]-1-cyclopropanecarbonylpiperidine-3-carboxylate
6-chloro-3-({4-[hydroxy(phenyl)methyl]piperidin-1-yl}methyl)-N,N-dimethylimidazo[1,2-a]pyridine-2-carboxamide
2-{2-[3-(acetamidomethyl)piperidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
2-[4-(2-amino-5-butyl-6-methylpyrimidin-4-yl)piperazin-1-yl]pyridine-3-carboxamide
4-{3-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine-5-carboxylic acid
1-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-1-methyl-3-propylurea
N-[(3R,4S)-4-cyclopropyl-1-(oxan-4-yl)pyrrolidin-3-yl]-1-ethyl-1H-pyrazole-4-carboxamide
methyl 5-[(1-acetylpiperidin-4-yl)amino]-1-(2-methoxyethyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(3S,4R)-4-methyl-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidine-3,4-diol
methyl 4-(5-methyl-4-{[(1S,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl}-1,3-oxazol-2-yl)benzoate
4-{[4-(propan-2-yl)phenyl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
2-(4-amino-1H-pyrazol-1-yl)-N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]acetamide
(3R,4R)-1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-3,4-dimethylpyrrolidin-3-ol
N3-(cyclohexylmethyl)-N5-(2-methoxyethyl)-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-methoxy-2-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,4-dihydropyridin-4-one
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-4-methoxybenzamide
5-(3-fluorophenyl)-3-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-1,2,4-triazine
6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-1,4-diazepan-2-one
N-[3-(3-oxopiperazin-1-yl)propyl]-3-propyl-1H-pyrazole-5-carboxamide
N-{1-cyclopentyl-7-[4-(pyridin-4-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl}benzamide
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}acetamide
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-[4-(morpholine-4-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
2-[2-(5-methoxypyridin-3-yl)phenoxy]propanamide
N-[4-({4-[(4-fluorophenyl)methyl]-5-oxo-1,4-diazepan-1-yl}methyl)phenyl]acetamide
N-[(2,5-dimethoxyphenyl)methyl]-1-(4,7-dimethylquinazolin-2-yl)piperidine-3-carboxamide
N-(2-methoxyethyl)-1-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-(quinolin-3-ylmethyl)-1H-pyrazole-4-carboxamide
N-phenyl-1-(thian-4-yl)piperidin-3-amine
1-[7-(1,3-benzothiazol-2-yl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-cyclopentylethan-1-one
7-[6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-3-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-propyl-6-[(thiophen-2-ylmethyl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
N,N-dimethyl-5-{[(1R,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyridin-2-amine
N-(1-methoxypropan-2-yl)-6-methyl-2-(4-methylphenoxymethyl)-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
4-[(4-fluorophenyl)methyl]-1-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)acetyl]-3-(propan-2-yl)-1,4-diazepan-5-one
[2-(1H-imidazol-1-yl)-1-phenylethyl]({[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl})amine
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}acetamide
N-[(3-chloro-4-fluorophenyl)methyl]-1-cyclopentanecarbonylpiperidine-4-carboxamide
2-{[(1r,4r)-4-hydroxycyclohexyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
(1R,5R)-6-(cyclopropylmethyl)-3-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
2-fluoro-N-(3-methoxypropyl)-N-{[6-(thiophen-2-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}benzamide
4-[(7-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]morpholine-2-carboxamide
4-[5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]-1-(oxan-4-yl)piperidine
5-fluoro-4-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]quinazoline
2,6-difluoro-3-methoxy-N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}benzamide
2-(3-chlorophenoxy)-1-[7-(1-hydroxy-2-methylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
2-[(1-methyl-2-oxopyrrolidin-3-yl)amino]pyridine-3-carboxamide
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine