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1-[3-(phenylamino)piperidin-1-yl]ethan-1-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
N-[3-(4-chlorophenyl)propyl]-1-cyclopentyl-5-oxopyrrolidine-3-carboxamide
(3aR,6aR)-2-(4-acetylbenzoyl)-5-(cyclobutylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[3-(3-fluorophenyl)phenyl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)piperidin-4-amine
(1R,5S)-6-{[5-(5-methylpyrazine-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-6-azabicyclo[3.2.1]octane
methyl 6-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-(1H-indol-1-ylmethyl)-N-[(3S)-2-oxoazepan-3-yl]-1H-pyrazole-3-carboxamide
2-fluoro-6-(1,2,3,4-tetrahydroisoquinolin-5-yl)benzamide
2-(4-ethyl-5-methylthiophene-3-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-5-methylthiophene-2-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(2-methylpyrimidine-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-(methoxymethyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}furan-2-carboxamide
4-[3-(3-methoxypiperidine-1-carbonyl)phenoxy]-N,N-dimethylpiperidine-1-sulfonamide
5-(5-methylfuran-2-yl)-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1,2,4-triazin-3-amine
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(6-methylpyridin-2-yl)piperazine
N-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-1H-1,2,3-triazol-4-amine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-methoxy-4-oxo-4H-pyran-2-carboxamide
1-tert-butyl-N-[2-(2-chloro-6-fluorophenyl)ethyl]-5-oxopyrrolidine-3-carboxamide
4-(1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)pyridine
5-methyl-2-(5-methylthiophen-2-yl)-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1,3-oxazole
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
5-benzenesulfonamido-1-ethyl-2-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
ethyl 1-(2-chloro-4-fluorobenzenesulfonyl)-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
N-(2-{5,6-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-2-yl}ethyl)-5-propyl-1,2-oxazole-3-carboxamide
2-[(4-benzylpiperazin-1-yl)methyl]-N-[2-(cyclohex-1-en-1-yl)ethyl]-1,3-oxazole-4-carboxamide
1-ethyl-N-methyl-2-oxo-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1,2-dihydropyridine-4-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-amine
N-[(2-ethoxypyridin-3-yl)methyl]-1-(oxan-4-yl)piperidine-4-carboxamide
1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
1-(1-benzothiophene-2-carbonyl)-4-(1-ethyl-1H-imidazol-2-yl)piperidine
4-({4-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]furan-2-yl}methyl)morpholine
N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
1-[1-(1,3-dihydroxypropan-2-yl)piperidin-3-yl]-2-phenylethan-1-one
4-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-1-phenylpiperidine
(1R,5R)-10-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-3,7,10-triazatricyclo[3.3.3.01,5]undecane-2,6-dione
5-(7-fluoro-1-methyl-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)quinoxaline
2-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-N-cyclopropylacetamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
N-ethyl-6-(4-methyl-1,4-diazepan-1-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
1-(2-{[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)amino}pyrimidin-4-yl)piperidin-3-ol
2-(3-methoxypropyl)-8-(quinolin-4-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)[(3-methoxyphenyl)methyl]amine
4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-7-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{1-[4-(2-ethylphenyl)piperazin-1-yl]-2-methyl-1-oxopropan-2-yl}thiophene-2-carboxamide
(4aR,7aS)-1-propyl-4-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{4-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]piperazin-1-yl}pyrazine
1-methyl-N-[2-(methylsulfanyl)phenyl]-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
2-fluoro-N-[3-methyl-1-(pyridin-3-yl)butyl]-5-sulfamoylbenzamide
3-(methanesulfonylmethyl)-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-1-carboxamide