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2-{[1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]formamido}-N,N-dimethylacetamide
1-[(5-ethylpyridin-2-yl)methyl]-3-(2-methoxy-6-methylphenyl)-1-methylurea
1-(3-{[(quinoxalin-2-yl)amino]methyl}pyridin-2-yl)piperidin-3-ol
4-{[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
1-ethyl-N-[(3R,4R)-4-hydroxypiperidin-3-yl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-(furan-2-yl)-N-(2-hydroxyethyl)-N-methyl-1H-pyrazole-4-carboxamide
N-[2-(4-fluorophenyl)-1-{1-[3-(thiophen-2-yl)propanoyl]piperidin-4-yl}ethyl]-2-methoxy-N-methylacetamide
N-[(2R,3R)-2-ethoxy-1'-[(2S)-2-hydroxy-2-phenylacetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-2-(4-methanesulfonylphenyl)ethan-1-one
1-[5-(4-cyclopentyl-1,4-diazepane-1-carbonyl)-2-methylphenyl]imidazolidin-2-one
1-(4-{[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-3-(1H-indol-3-yl)propan-1-one
3-(hydroxymethyl)-N-(4-methoxy-2-methylphenyl)piperidine-1-carboxamide
N-(5-chloropyridin-2-yl)-4-{[methyl(oxolan-2-ylmethyl)amino]methyl}benzamide
ethyl 2-{1-[3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanoyl]piperidin-2-yl}acetate
2-cyclopropyl-1-[(4-fluorophenyl)methyl]-6-methyl-3-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(morpholin-4-yl)propyl]acetamide
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-3-{[5-(pyridin-4-yl)-1,3,4-oxadiazol-2-yl]sulfanyl}propan-1-one
N4,N4,5-trimethyl-N2-[1-(pyrimidin-4-yl)ethyl]pyrimidine-2,4-diamine
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-(4-hydroxypiperidin-1-yl)pyridine-3-carboxamide
2-amino-4-{4-[(dimethylamino)methyl]thiophen-2-yl}-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
2,6-di-tert-butyl-4-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenol
N-[3-(pyridin-4-yl)propyl]-2-(trifluoromethyl)pyrimidin-4-amine
ethyl 4-{[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]amino}piperidine-1-carboxylate
2-{1-[(3,4-difluorophenyl)methyl]-4-[(2-fluoro-5-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
(2S)-4-carbamoyl-2-[4-phenyl-5-(propan-2-yl)-1H-imidazol-1-yl]butanoic acid
N-cyclopentyl-N'-(2,2-diphenylethyl)butanediamide
8-[2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)acetyl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
7-chloro-4-(5-methyl-1,3,4-oxadiazol-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[2-(4-chlorophenyl)ethyl]-5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}dimethylamine
N-{[3-cyclopropyl-1-(3-methylphenyl)-1H-1,2,4-triazol-5-yl]methyl}-N,1-dimethylpiperidin-4-amine
(1S,5R)-6-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-(2-ethoxyphenyl)-3-(1-methyl-1H-pyrazol-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,5R)-1-[(2-methoxyphenyl)methyl]-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
(2E)-3-(1H-imidazol-4-yl)-N-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}prop-2-enamide
8-(cyclohex-3-en-1-ylmethyl)-1-(2-methoxyethyl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[2-(2-methoxyethoxy)acetyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
4-{4-[(3S)-3-(dimethylamino)pyrrolidin-1-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}benzamide
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)butanamide
3-(4-chlorophenyl)-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-3-phenylpropanamide
3-(2-fluorophenyl)-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-phenylpropanamide
6-(3,4-dimethylpiperazin-1-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
1-(1-benzofuran-2-carbonyl)-4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine
1-(2-{methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino}pyrimidin-4-yl)pyrrolidin-3-ol
1-(4-fluorophenyl)-2,2-dimethyl-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)cyclopropane-1-carboxamide
6-(2,4,6-trimethylphenyl)pyridin-2-amine
5-ethyl-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)thiophene-2-carboxamide
4-cyclobutyl-N-{[3-(3-fluorophenyl)-1,2-oxazol-5-yl]methyl}-6-methylpyrimidin-2-amine
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propan-1-one
2-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-7-propyl-2,7-diazaspiro[4.5]decan-6-one