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(2S,4S)-N-ethyl-4-{[(2E)-2-methylbut-2-en-1-yl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
4-benzyl-1-methyl-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-ethyl-1-({4-[(1,2,3-thiadiazol-5-yl)carbamoyl]phenyl}methyl)pyrrolidine-3-carboxamide
1-cyclohexyl-4-oxo-5-(pyrrolidine-1-carbonyl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
3,4,7-trimethyl-2-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carbonyl}-1H-indole
2-(4-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-(1-methylpiperidin-4-yl)piperazin-2-yl)ethan-1-ol
ethyl 3-[(4-fluorophenyl)methyl]-1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidine-3-carboxylate
2-amino-4-[methyl({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl})amino]quinazoline-6-carboxylic acid
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]pyrazolo[1,5-a]pyridine-7-carboxamide
(1R,5S)-8-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,8-diazabicyclo[3.2.1]octane
N-(2-chlorophenyl)-2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxamide
ethyl 5-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-1-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(2-hydroxybutyl)-5-methyl-4-{[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
1-[3-(3-chlorophenyl)pyrrolidin-1-yl]-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}ethan-1-one
3-propoxy-1-(1,2,3,4-tetrahydronaphthalen-2-yl)piperidine
6-{[(1-carbamoylethyl)(methyl)amino]methyl}-2-oxo-N-(quinolin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
1-methyl-3-{2-oxo-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl}-3-(4-phenylphenyl)pyrrolidine-2,5-dione
3-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(isoquinolin-5-yl)urea
6-methyl-N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazole-4-carboxamide
1-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-2-(methoxymethyl)piperidine
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-methoxy-2-methylpropan-1-one
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
[(6-chloropyridin-3-yl)methyl](ethyl)(oxolan-2-ylmethyl)amine
2-methyl-4-[5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)furan-2-yl]but-3-yn-2-ol
(1S,5R)-3-(1-benzothiophen-2-ylmethyl)-3,9-diazabicyclo[3.3.2]decan-10-one
N-(cyclohex-1-en-1-ylmethyl)-2-(propan-2-yl)pyrimidine-5-carboxamide
1-[1-(3-chloro-4-fluorobenzoyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
(2S,4R)-4-(4-{[1-(2,3-difluorophenyl)-N-methylformamido]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
4-[(4-methyl-5-{[(2,4,5-trifluorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]piperidine
N-cyclohexyl-2-methyl-N-(pyridin-4-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
N-(oxan-4-ylmethyl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
1-cyclohexyl-N-(cyclopropylmethyl)-N-propyl-1H-1,2,3-triazole-4-carboxamide
1-(4-methoxyphenyl)-4-[2-(2-methylpyrrolidin-1-yl)-2-oxoethyl]-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(3aR,5R,6S,7aS)-2-(2,2-diphenylethyl)-octahydro-1H-isoindole-5,6-diol
3-[5-(3-ethyl-4-methyl-1H-pyrazol-5-yl)-1,2,4-oxadiazol-3-yl]pyridazine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(morpholin-3-yl)acetamide
methyl 5-[(4-hydroxy-4-methylpentan-2-yl)amino]-1-methyl-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[2-(4-fluorophenyl)pyrrolidin-1-yl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
2-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-N-(prop-2-en-1-yl)pyridine-3-carboxamide
4-({5-[(dimethyl-1,3-thiazol-4-yl)methyl]-1,2,4-oxadiazol-3-yl}methyl)-1-methylpiperidine
N-[2-(1H-imidazol-1-yl)propyl]-1,3,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl 5-(3-phenoxypropanoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
1-methyl-N-(pyridin-3-ylmethyl)-5-{[4-(trifluoromethoxy)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-chloro-N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
4-[(4-chloro-2-fluorophenyl)methyl]-2-ethyl-1-(propan-2-yl)piperazine
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-4-phenylbutanamide
2-(5-fluoro-2-methylphenyl)-1-[2-(2-hydroxyethyl)morpholin-4-yl]ethan-1-one
(3S)-3-ethyl-4-[4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carbonyl]morpholine