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N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-benzyl-4-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]morpholine
4-ethyl-3-(piperidin-4-yl)-1-[2-(1H-1,2,4-triazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(3aS,6aS)-2-methyl-5-(5-methyl-1,3,4-thiadiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
7-methoxy-N,4-dimethyl-N-[2-(morpholin-4-yl)propyl]quinazolin-2-amine
5-ethyl-3-(2-methylprop-2-en-1-yl)-5-[1-(1-phenyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
4-[1-(2-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,3-thiazole
1-(2-phenylethyl)-3-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3aS,6aS)-2-[(dimethyl-1,3-thiazol-5-yl)methyl]-5-(ethanesulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)pent-4-enamide
(2S,4R)-N-(diphenylmethyl)-1-[(4-methoxynaphthalen-1-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[(3-methylphenyl)methyl]piperidine
3-butyl-1-methyl-4-[4-(piperidin-1-yl)benzoyl]piperazin-2-one
4-cyano-N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)oxane-4-carboxamide
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-methoxypyridine-3-carbonitrile
3-({[3-(2,4-dimethylphenoxy)propyl](methyl)amino}methyl)piperidin-3-ol
methyl[3-(morpholin-4-yl)propyl]({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(2H-1,3-benzodioxol-5-ylmethyl)({[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
(3aS,6aS)-2-(cyclopropylmethyl)-5-[(2,3-difluoro-4-methylphenyl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(4-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-4-oxobutyl)pyrrolidin-2-one
2-(1H-pyrazol-1-yl)-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]butanamide
N-cyclopentyl-4-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]benzamide
2-(4-{[2-(cyclopentyloxy)phenyl]methyl}-1-(1-methylpiperidin-4-yl)piperazin-2-yl)ethan-1-ol
3-{2-oxo-2-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]ethyl}-1,3-oxazolidin-2-one
ethyl 1-{[3-(furan-2-amido)-2-(methoxycarbonyl)thieno[2,3-b]pyridin-6-yl]methyl}piperidine-4-carboxylate
2-[7-(hydroxymethyl)-9-(2-methoxyethyl)-3,9-diazaspiro[5.5]undecan-3-yl]acetic acid
2-(1-{5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-4-yl)ethan-1-ol
N-(4-{1-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1H-imidazol-2-yl}phenyl)acetamide
N-methyl-N-{1-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-2-phenylethyl}thiophene-2-carboxamide
3-(2-hydroxy-1-phenylethyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1-benzothiophene-2-carboxamide
[2-(2,6-dimethylphenoxy)ethyl](ethyl)(1,3-thiazol-2-ylmethyl)amine
5-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-6-methylimidazo[2,1-b][1,3]thiazole
2-[4-(dimethylamino)phenyl]pyridine-4-carboxamide
4-{2-[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]-1-(pyridin-2-yl)ethyl}morpholine
[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl})amine
(3S,4S)-1-[3-(dimethylamino)-1,2,4-thiadiazol-5-yl]-4-methylpiperidine-3,4-diol
1'-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
N-[(5-methylfuran-2-yl)methyl]-3-{1-[3-(prop-2-en-1-yloxy)benzoyl]piperidin-3-yl}propanamide
3,5-dichloro-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-4-methylbenzamide
{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
1-[1-(oxane-4-carbonyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
5-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-3-[(2,3-dimethoxyphenyl)methyl]-5-methylimidazolidine-2,4-dione
2-{2-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]acetamido}-N-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
1-[3-(azocane-1-carbonyl)benzenesulfonyl]piperidin-3-ol
N-{2-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]propan-2-yl}aniline
5-propyl-1'-{thieno[3,2-d]pyrimidin-4-yl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(4-fluorophenyl)methyl]-5-[1-(methoxymethyl)cyclobutyl]-1H-1,2,4-triazole