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4-{[2-(dimethylamino)ethyl]amino}-5-methyl-N-[2-(methylsulfanyl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
2-(benzyloxy)-1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]ethan-1-one
{1-[(2-fluoro-5-methylphenyl)methyl]-3-(3-methoxypropyl)piperidin-3-yl}methanol
2-amino-6-(1-ethyl-1H-indol-3-yl)-4-(4-methyl-1H-imidazol-5-yl)pyridine-3-carbonitrile
2-{1-[(4-ethoxyphenyl)methyl]-4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
1-[(2S,4S)-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carbonyl]-4-phenylpiperazine
4-(cyclopropylmethyl)-1-[(3,4-dimethoxypyridin-2-yl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-benzyl-8-(2,3-dihydro-1H-inden-2-yl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-methoxy-3,5-dimethylphenyl)-2-[4-(2-methoxyethoxy)piperidin-1-yl]acetic acid
(3S)-4-{2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-1-ethyl-3-methylpiperazin-2-one
N-[(2-fluorophenyl)methyl]-1-{2-[2-(2-methoxyphenyl)acetamido]ethyl}-1H-1,2,3-triazole-4-carboxamide
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-(1,4-oxazepan-4-ylmethyl)piperidin-2-one
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(1-methoxybutan-2-yl)acetamide
4-[3-(2-hydroxyethyl)-4-(1-methylpiperidin-4-yl)piperazin-1-yl]-2-methoxypyridine-3-carbonitrile
3-(5-methylfuran-2-yl)-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-1H-pyrazole-5-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-cyclobutyl-5-(2-methoxyacetamido)-N,1-dimethyl-1H-1,3-benzodiazole-7-carboxamide
1-cyclohexyl-N3-cyclopropyl-4-oxo-N5-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(5-{[4-(4-phenyl-1,3-thiazol-2-yl)piperazin-1-yl]methyl}furan-2-yl)methanol
2-cyclopentyl-N-[3-(4-{[2-(pyridin-4-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
N-(5-fluoro-2-methoxyphenyl)-2-(2-hydroxyethyl)pyrrolidine-1-carboxamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(4-ethylphenyl)methyl]-5-methoxy-N-methylbenzamide
N-{[(2S,4S)-4-fluoro-1-[(4-methoxy-5,6,7,8-tetrahydronaphthalen-1-yl)sulfonyl]pyrrolidin-2-yl]methyl}acetamide
(3S,4S)-1-(1H-imidazol-4-ylmethyl)-4-[4-(2-methylphenyl)-1,4-diazepan-1-yl]pyrrolidin-3-ol
5-({[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}methyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
5-{2-[4-(2-methoxyethyl)phenoxymethyl]phenyl}pyrazin-2-amine
2-[2-(1H-imidazol-4-yl)ethyl]-8-[2-(pyridin-3-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
9-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-methoxypyrimidine-5-carboxamide
2-[2-(benzyloxy)phenyl]-1-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-[2-(1,3,4-oxadiazol-2-yl)phenyl]-1-(oxolan-2-ylmethyl)-1-(pyridin-2-ylmethyl)urea
3-[2-(2,5-dihydro-1H-pyrrol-1-yl)-2-oxoethyl]-5-methyl-2,3-dihydro-1H-indol-2-one
4-{1-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]pyrrolidin-3-yl}-2-(pyridin-4-yl)pyridine
1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]-2-(4,6,7-trimethyl-1-benzofuran-3-yl)ethan-1-one
2-(4-{1-[3-(methylsulfanyl)propyl]pyrrolidin-3-yl}piperidin-1-yl)pyrimidine
3-(4-methoxyphenyl)-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]-1H-pyrazole-5-carboxamide
methyl 6-[(oxan-2-ylmethyl)carbamoyl]pyridine-3-carboxylate
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
ethyl 1-benzyl-5-[1-(pyridin-2-yl)piperidine-3-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-[3-(3-fluorophenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-(2-methoxyethyl)-N-methylacetamide
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}acetamide
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-4-(piperidin-1-ylmethyl)benzamide
N-{[2-(4-chlorophenyl)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-1,3-thiazole-5-carboxamide
[(5-methoxy-1,3-benzoxazol-2-yl)methyl]({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
1-ethyl-4-(5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)piperazine
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-1-[2-(3-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
5-chloro-3-methyl-2-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}methyl)-1H-indole
3-{[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenol
3-(furan-2-yl)-1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}propan-1-one