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2-[4-({[(4,6-dimethylpyridin-2-yl)methyl](methyl)amino}methyl)-2-methoxyphenoxy]propanoic acid
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-ethylpyrimidine
N-methyl-2-({3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}sulfanyl)-N-[(4-phenoxyphenyl)methyl]acetamide
1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-(1,2-oxazol-3-ylmethyl)piperidine-3-carboxamide
(3aR,6aS)-5-[(6-ethoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]propane-1-sulfonamide
N-[6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-1-propylpiperidin-4-amine
11-{[(2,6-difluorophenyl)methyl]amino}-4-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-{[1-cyclohexyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-4-ethylpiperazin-2-one
[1-({[(2-fluoro-3-methoxyphenyl)methyl](methyl)amino}methyl)cyclopropyl]methanol
3-{4-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-yl}pyridine
3-benzyl-4-(2,5-difluorobenzoyl)piperazin-2-one
4-(3,6-dimethylpyrazin-2-yl)-2-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenol
1-[1-(3-methylpyrazin-2-yl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]benzamide
N-{[7-(3,5-dimethylbenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
3-[(propan-2-yl)sulfamoyl]-5-(1H-pyrazol-3-yl)benzoic acid
ethyl 1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
(1R,5R)-N,N-dimethyl-6-(6-methylpyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
3-[4-(3-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)piperidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-3-[5-oxo-2-(thiophen-3-ylmethyl)pyrrolidin-2-yl]propanamide
1-phenyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1H-1,2,3-triazole-5-carboxamide
2-[4-(3-aminophenyl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
1-(2-fluorophenyl)-4-[1-(3-methoxybenzoyl)piperidin-3-yl]piperazine
4-(3-chlorobenzoyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(2R,3R)-3-[(2H-1,3-benzodioxol-5-ylmethyl)(methyl)amino]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-cycloheptyl-1-{4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}ethan-1-one
4-hydroxy-2-(4-methylphenyl)-N-[(2-propyl-1,3-thiazol-4-yl)methyl]pyrimidine-5-carboxamide
(2S,4S)-N-methyl-4-{4-[(2-phenylacetamido)methyl]-1H-1,2,3-triazol-1-yl}pyrrolidine-2-carboxamide
N-(2-methoxyethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
(1R,5R)-N,N-dimethyl-6-(5,6,7,8-tetrahydroquinoline-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[4-(4-{[1-(1,3-thiazol-5-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]-2H-1,3-benzodioxole-5-carboxamide
N-cyclopropyl-N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)-2-(trifluoromethoxy)benzene-1-sulfonamide
N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-N'-(2-fluoro-5-methylphenyl)butanediamide
3-({ethyl[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)pyridin-2-amine
1-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)-2-[(2-methylphenyl)sulfanyl]ethan-1-one
(2R,3R)-3-amino-1'-(4-ethyl-5-methylpyrimidin-2-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[1-(1-{[2-(5-methylfuran-2-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]acetamide
2-amino-6-(6-methoxypyridin-3-yl)-4-(oxolan-3-yl)pyridine-3-carbonitrile
1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
(3R,4S)-4-[(2,2-diphenylethyl)(methyl)amino]oxolan-3-ol
1-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-3-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]urea
N-(2-oxo-4-{pyrazolo[1,5-a]pyrimidin-3-yl}-1,2,3,4-tetrahydroquinolin-7-yl)methanesulfonamide
N-(2-hydroxybutyl)-4-[methyl(1,2-oxazol-3-ylmethyl)sulfamoyl]benzamide
N-{[7-(2,2,3,3-tetramethylcyclopropanecarbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}oxolane-3-carboxamide
1-(5-chloro-2-methylphenyl)-4-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
2-({[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]({[2-(2-methylphenoxy)pyridin-3-yl]methyl})amine
N-ethyl-2-[N-(3-fluorophenyl)methanesulfonamido]-N-(pyridin-4-ylmethyl)acetamide