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6-(3-fluorophenyl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
2-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]quinoxaline
3-(1-{[5-(2-chlorophenyl)furan-2-yl]methyl}piperidin-3-yl)-N-cyclopropylpropanamide
1-[1-(1,4-dithiepan-6-yl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
3-(3,4-dimethoxybenzoyl)-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]piperidine
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-phenoxybutan-1-one
2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(4aS,8aS)-2-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-decahydroisoquinolin-4a-ol
[4-(oxan-2-ylmethyl)-1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-4-yl]methanol
{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(3,4-dimethoxyphenyl)methyl]methylamine
methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)[(2E)-3-phenylprop-2-en-1-yl]amine
5-{1-[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}-2-(furan-2-yl)pyrimidine
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(2H-1,3-benzodioxol-5-yl)-1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}propan-1-one
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-(2-phenylethyl)-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
5-[(3-fluorophenyl)methyl]-3-(2-methoxyethyl)-5-{1-[2-(3-methoxyphenyl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
2-cyclohexyl-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,3-benzoxazole-6-carboxamide
3-ethyl-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1-methyl-1H-pyrazole-5-carboxamide
N,N-dimethyl-3-[5-(trifluoromethyl)-1H-1,2,4-triazol-3-yl]aniline
ethyl 1-[(4-acetamidophenyl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
4-{[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-(2-fluorophenyl)ethyl)piperidin-1-yl]methyl}-2-methoxyphenol
N-[2-(3-fluorophenyl)ethyl]-2-[4-(4-{[1-(pyridin-2-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]acetamide
1-{2H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-6-chloroimidazo[1,2-a]pyrimidine-2-carboxamide
5-cyclopropyl-N-[3-(dimethylamino)-2,2-dimethylpropyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-(1H-indol-3-ylmethyl)-2,7-diazaspiro[4.5]decane
2-({4-[(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)benzonitrile
(1R,6S)-3-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-9-methyl-3,9-diazabicyclo[4.2.1]nonane
methyl 8-[(2,6-difluorophenyl)methyl]-1-ethoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
(2R,3R,6R)-3-phenyl-5-(quinolin-5-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-cyclopentanecarbonyl-N-[(2-ethoxypyridin-3-yl)methyl]piperidine-4-carboxamide
1-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-2-methyl-2-(morpholin-4-yl)propan-1-one
(2R,3R,6R)-3-(4-fluorophenyl)-5-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-({[3-(4-fluorophenyl)propyl]carbamoyl}methyl)piperidine-4-carboxamide
1-[(3-chloro-4-hydroxyphenyl)methyl]-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
methyl 2-[(cyclohexylmethyl)sulfamoyl]-6-[(4-hydroxyphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-[3-(1,2-oxazolidin-2-yl)propanoyl]-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
6-(dimethylamino)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
(5S,9aS,9bS)-5-(4-fluoro-3-methoxyphenyl)-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-ethoxy-4-({3-[5-(2-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenol
3-hydroxy-1-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
ethyl 4-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}piperidine-1-carboxylate
2-[4-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-6-hydroxy-1,4-diazepan-1-yl]acetamide
butyl({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)methylamine
1-[(2-methylphenyl)methyl]-4-[3-(methylsulfanyl)propyl]piperazine
1-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)-2-(3,4-dimethoxyphenyl)-5-fluoro-1H-1,3-benzodiazole
methyl 1-[(3S,5S)-1-[(4-methoxy-3-methylphenyl)methyl]-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
(3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl){[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}amine