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N-{1-[4-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-1-oxopropan-2-yl}methanesulfonamide
2-(3-phenyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-{3-[({7-methylthieno[3,2-d]pyrimidin-4-yl}amino)methyl]pyridin-2-yl}piperidin-3-ol
1-[5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-3-(2-methylphenyl)piperidine
3-[1-(5-methoxyfuran-2-carbonyl)piperidin-3-yl]-1-(pyrrolidin-1-yl)propan-1-one
1-(4-fluorophenyl)-4-[4-(piperidin-3-yl)benzoyl]-1,4-diazepane
2-({4-[4-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
N2,N2-dimethyl-5,6,7,8-tetrahydroquinazoline-2,5-diamine
4-(cyclopropylmethyl)-1-(4,6-dihydroxypyridine-3-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
3-[1-(2-methyl-1-benzofuran-5-carbonyl)piperidin-4-yl]-1,3-oxazolidin-2-one
(4aR,8aS)-6-[(2,4-dimethoxy-3-methylphenyl)methyl]-1-(2-methoxyethyl)-decahydro-1,6-naphthyridin-2-one
N-{2-[(pyridin-3-yl)amino]ethyl}-2-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide
8-(5,6,7,8-tetrahydroquinoline-3-carbonyl)-1-oxa-8-azaspiro[4.6]undecane
2-[1-(4-chlorophenyl)-3-(furan-2-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-[(2S)-2-hydroxypropyl]acetamide
(3R,4S)-1-(5-methoxyfuran-2-carbonyl)-3,4-dimethylpiperidin-4-ol
methyl 5-[(2R,3R)-3-acetamido-2-(pyridin-4-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-5-oxopentanoate
N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-2-(pyridin-2-ylsulfanyl)acetamide
1-(2-oxo-2-{spiro[indene-1,4'-piperidine]-1'-yl}ethyl)-1,2-dihydropyrimidin-2-one
1-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-4-(morpholin-4-yl)butan-1-one
(3aR,5S,6S,7aS)-2-[(2-chlorophenyl)methyl]-octahydro-1H-isoindole-5,6-diol
5-(2,6-difluorophenoxymethyl)-N-methyl-N-(naphthalen-1-ylmethyl)-1,2-oxazole-3-carboxamide
N-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
[(3S,5R)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl]methanol
methyl 7-oxo-3-(2-oxo-2-phenylacetyl)-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3,4,7-trimethyl-2-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1H-indole
(1S,6R)-9-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
2-methoxy-5-({[(2R)-1,1,1-trifluoro-3-methylbutan-2-yl]carbamoyl}amino)benzamide
methyl 6-[4-(4-hydroxyphenyl)butan-2-yl]-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
methyl 6-oxo-4-[2-(propan-2-yl)pyrimidin-4-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylate
6-ethyl-2-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}quinoline-4-carboxamide
1-[3-(dimethylcarbamoyl)pyridin-2-yl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-[(2,3-difluorophenyl)methyl]-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}propane-1-sulfonamide
5-[2-(pyridin-4-yl)-1H-imidazol-1-yl]-1,3-benzothiazole
5-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]-3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propylimidazolidine-2,4-dione
N,N-dimethyl-5-({methyl[1-(3-methylpyridin-2-yl)propan-2-yl]amino}methyl)pyridin-2-amine
N-[(4-methoxypyridin-2-yl)methyl]-N-methyl-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
2-{[(1S)-1-(3-methylpyridin-2-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-amino-5-methyl-4-(1-methyl-1H-indol-6-yl)-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-(1-{[3-(cyclopentyloxy)phenyl]methyl}piperidin-4-yl)methanesulfonamide
1-[3-(3-methoxypropyl)piperidin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
6-{[3-(3-methylbutyl)-1,2,4-oxadiazol-5-yl]methoxy}-1,2-benzoxazole
N-[2-(2,3-dimethoxyphenyl)ethyl]-1-methylazepane-2-carboxamide
N-({7-[2-(3-methoxyphenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)ethane-1-sulfonamide
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]pyrazolo[1,5-a]pyridine-7-carboxamide
3-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]-1-(oxan-4-yl)urea
2-({5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)-1-(pyridin-3-yl)ethan-1-ol
methyl 3-(3-methylpentanoyl)-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(2S,4R)-4-amino-N-ethyl-1-[(2-methoxy-4-methylphenyl)methyl]pyrrolidine-2-carboxamide
4-{5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]benzoyl}thiomorpholine