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2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-(2-methoxy-2-methylpropyl)acetamide
methyl({[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}){[4-(propan-2-yl)phenyl]methyl}amine
N-[2-(cyclohexylsulfanyl)ethyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-1-methylazepane-2-carboxamide
9-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(4-methylphenyl)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
6-methyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
ethyl 1-{2-[1-cyclopentyl-3-(2-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]acetyl}piperidine-4-carboxylate
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-cyclopropylacetamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(2-fluoro-5-methylphenoxy)piperidine-4-carboxylic acid
3-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-1-[4-(1H-pyrazol-4-yl)phenyl]urea
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(9H-purin-6-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-(cyclopropylmethyl)-1-(8-methoxy-4-methylquinolin-2-yl)piperidine-4-carboxylic acid
N-ethyl-7-methoxy-N-methyl-2-[1-(pyridin-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
2-hydroxy-3-methyl-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)butanamide
5-[4-(aminomethyl)piperidin-1-yl]-2-[2-(2-methoxyphenoxy)ethyl]-2,3-dihydropyridazin-3-one
2-cyclopropyl-1-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
(4aS,7aR)-1-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2-phenylethyl)-9-[(1-propyl-1H-imidazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}morpholin-3-yl)acetic acid
3-methyl-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]benzamide
3-{2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}-5,6-dimethyl-1,2-dihydropyridin-2-one
2-{2-oxo-2-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethyl}-1,2-dihydrophthalazin-1-one
(3S,9aR)-3-[(2S)-butan-2-yl]-8-(3,5-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]pyrazin-2-amine
N-methyl-N-[(5-methylfuran-2-yl)methyl]-4H-thieno[3,2-b]pyrrole-5-carboxamide
5-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-3-(cyclopropylmethyl)-5-[(4-fluorophenyl)methyl]imidazolidine-2,4-dione
2-(1H-imidazol-1-yl)-1-[3-(4-methylphenoxymethyl)piperidin-1-yl]ethan-1-one
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-decahydro-1,6-naphthyridin-2-one
2-fluoro-6-({4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)phenol
2-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine-1-carbonyl)-1H-indole
3-(3,5-dimethyl-4-{4-[1-(piperidin-1-yl)ethyl]phenyl}-1H-pyrazol-1-yl)propanamide
1-cyclohexyl-4-(5-methyl-1H-indazole-3-carbonyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
4-(4-{1-[4-(1H-1,2,3,4-tetrazol-5-yloxy)phenyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-6-hydroxy-N-(oxolan-2-ylmethyl)pyridine-3-carboxamide
1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(2-phenylethyl)piperidine
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-methyloxane-2-carboxamide
(2S,4R)-1-[(2-hydroxy-4-methoxyphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-[2-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
3-(1H-1,3-benzodiazol-2-yl)-1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
4-(5-methylpyridin-2-yl)-1-[6-(trifluoromethyl)pyridin-2-yl]piperidin-4-ol
4-{2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-4-oxobutanamide
4-[(2-fluoro-4-methoxyphenyl)methyl]-3-{2-[4-(morpholin-4-yl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
1-[(2-propylpyrimidin-5-yl)methyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
5-(1-benzofuran-2-yl)-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1,2,4-triazin-3-amine
1-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-3-[(1-methyl-1H-imidazol-2-yl)methyl]-3-propylurea
9-methoxy-7-(6-methoxypyridin-2-yl)-4-(naphthalen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(5-methylpyrazin-2-yl)methyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide